SCHEMBL408023

SCHEMBL408023

CN(c1ncccc1CN)S(C)(=O)=O

nearest known ligand 0.54

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTK2 Q05397 14/20 0.54
SRPK1 Q96SB4 5/20 0.45
PTK2B Q14289 1/20 0.43
SRPK2 P78362 4/20 0.42
SRPK3 Q9UPE1 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL30468512 0.98 PTK2 (0.53) PTK2SRPK1PTK2BSRPK2SRPK3
Hydrochloric Acid SCHEMBL29051922 0.98 PTK2 (0.53) PTK2SRPK1PTK2BSRPK2SRPK3
Acetic Acid SCHEMBL1627284 0.93 PTK2 (0.49) PTK2SRPK1PTK2B
SCHEMBL10229210 0.87 PTK2 (0.53) PTK2SRPK1PTK2BSRPK2SRPK3
Methane SCHEMBL4887418 0.86 PTK2 (0.44) PTK2SRPK1PTK2BSRPK2SRPK3
SCHEMBL16569929 0.85 PTK2 (0.52) PTK2SRPK1PTK2BSRPK2SRPK3
SCHEMBL16570123 0.84 PTK2 (0.51) PTK2SRPK1PTK2BSRPK2SRPK3
SCHEMBL17993894 0.83 PTK2 (0.40) PTK2SRPK1SRPK2
SCHEMBL1291246 0.81 ALDH1A1 (0.39) PTK2SRPK1
SCHEMBL12586298 0.81 PTK2 (0.58) PTK2SRPK1PTK2BSRPK2SRPK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 117 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118852119-A Light affinity probe for targeting local focal adhesion kinase and preparation method and application thereof 南京科络思生物科技有限公司 2024-10-29 CN claimed
CN-118852119-A Light affinity probe for targeting local focal adhesion kinase and preparation method and application thereof 南京科络思生物科技有限公司 2024-10-29 CN disclosed
CN-118852119-A Light affinity probe for targeting local focal adhesion kinase and preparation method and application thereof 南京科络思生物科技有限公司 2024-10-29 CN disclosed
US-11981665-B2 Substituted pyrimidines, pharmaceutical compositions and therapeutic methods thereof CHEN ZHIHONG (US) 2024-05-14 US disclosed
CN-111683662-B Substituted pyrimidine compounds, pharmaceutical compositions and methods of treatment 陈志宏 2024-04-02 CN disclosed
US-20230109688-A1 SUBSTITUTED PYRIMIDINES, PHARMACEUTICAL COMPOSITIONS AND THERAPEUTIC METHODS THEREOF CHEN ZHIHONG (US) 2023-04-13 US disclosed
EP-3675860-B1 SUBSTITUTED PYRIMIDINES, PHARMACEUTICAL COMPOSITIONS AND THERAPEUTIC METHODS THEREOF ZHIHONG CHEN (US) 2023-03-08 EP disclosed
US-11440904-B2 Substituted pyrimidines, pharmaceutical compositions and therapeutic methods thereof CHEN ZHIHONG (US) 2022-09-13 US disclosed
CN-111683662-A Substituted pyrimidines, pharmaceutical compositions and methods of treatment 陈志宏 2020-09-18 CN disclosed
EP-3675860-A1 SUBSTITUTED PYRIMIDINES, PHARMACEUTICAL COMPOSITIONS AND THERAPEUTIC METHODS THEREOF Zhihong, Chen (US) 2020-07-08 EP disclosed
WO-2009071535-A1 DIAMINOPYRIDINES FOR THE TREATMENT OF DISEASES WHICH ARE CHARACTERISED BY EXCESSIVE OR ANOMAL CELL PROLIFERATION BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-06-11 WO disclosed
US-20090054395-A1 SULFONYL AMIDE DERIVATIVES FOR THE TREATMENT OF ABNORMAL CELL GROWTH PFIZER INC. 2009-02-26 US disclosed
US-20090054395-A1 SULFONYL AMIDE DERIVATIVES FOR THE TREATMENT OF ABNORMAL CELL GROWTH PFIZER INC. 2009-02-26 US disclosed
CN-101346380-A Pyrimidine derivatives for the treatment of abnormal cell growth PFIZER PROD INC (US) 2009-01-14 CN disclosed
WO-2008129380-A1 SULFONYL AMIDE DERIVATIVES FOR THE TREATMENT OF ABNORMAL CELL GROWTH PFIZER PRODUCTS INC. (US) 2008-10-30 WO disclosed
US-20080234303-A1 PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF ABNORMAL CELL GROWTH PFIZER INC 2008-09-25 US disclosed
WO-2008115369-A2 INHIBITORS OF FOCAL ADHESION KINASE THE SCRIPPS RESEARCH INSTITUTE (US) 2008-09-25 WO disclosed
WO-2008115369-A2 INHIBITORS OF FOCAL ADHESION KINASE THE SCRIPPS RESEARCH INSTITUTE (US) 2008-09-25 WO disclosed
EP-1966207-A2 PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF ABNORMAL CELL GROWTH Pfizer Products Inc. (US) 2008-09-10 EP disclosed
WO-2007072158-A2 PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF ABNORMAL CELL GROWTH PFIZER PRODUCTS INC. (US) 2007-06-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080234303-A1 PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF ABNORMAL CELL GROWTH CCNB1, TYMS, CCNA1 PTK2 2406/4885SRPK1 218/4885PTK2B 1390/4885
US-20230109688-A1 SUBSTITUTED PYRIMIDINES, PHARMACEUTICAL COMPOSITIONS AND THERAPEUTIC METHODS THEREOF BTK, PTK2, LCK PTK2 2/4885SRPK1 643/4885PTK2B 7/4885
US-20090054395-A1 SULFONYL AMIDE DERIVATIVES FOR THE TREATMENT OF ABNORMAL CELL GROWTH GPR119, INSR, LYAR PTK2 4052/4885SRPK1 518/4885PTK2B 3523/4885
US-11981665-B2 Substituted pyrimidines, pharmaceutical compositions and therapeutic methods thereof BTK, PTK2, LCK PTK2 2/4885SRPK1 643/4885PTK2B 7/4885
US-11440904-B2 Substituted pyrimidines, pharmaceutical compositions and therapeutic methods thereof BTK, PTK2, LCK PTK2 2/4885SRPK1 643/4885PTK2B 7/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.