Triaziquone

Triaziquone

SCHEMBL4082601

CC(P)C(=O)O.O=C1C=C(N2CC2)C(=O)C(N2CC2)=C1N1CC1

nearest known ligand 0.39

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DNMT1 P26358 1/20 0.39
MAPT P10636 2/20 0.37
TP53 P04637 1/20 0.37
STAT3 P40763 1/20 0.37
HTT P42858 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
APAF1 O14727 2/20 0.33
TDP2 O95551 2/20 0.33
NSD2 O96028 2/20 0.33
HKDC1 Q2TB90 2/20 0.33
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
GALK1 P51570 1/20 0.32
BLM P54132 1/20 0.32
ATM Q13315 1/20 0.32
NOD2 Q9HC29 1/20 0.32
ATG4B Q9Y4P1 1/20 0.32
DHODH Q02127 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Triaziquone SCHEMBL11583629 0.90 DNMT1 (0.41) DNMT1MAPTTP53STAT3HTT
Triaziquone SCHEMBL6535620 0.89 DNMT1 (0.40) DNMT1MAPTTP53STAT3HTT
Triaziquone SCHEMBL5803947 0.89 DNMT1 (0.42) DNMT1MAPTTP53STAT3HTT
Triaziquone SCHEMBL112498 0.88 DNMT1 (0.39) DNMT1MAPTTP53STAT3HTT
Triaziquone SCHEMBL16419 0.85 MAPT (0.42) DNMT1MAPTTP53STAT3HTT
Triaziquone SCHEMBL7925866 0.85 DNMT1 (0.37) DNMT1MAPTTP53STAT3HTT
Triaziquone SCHEMBL4608905 0.85 DNMT1 (0.43) DNMT1MAPTTP53STAT3HTT
Triaziquone SCHEMBL7567124 0.84 DNMT1 (0.41) DNMT1MAPTTP53STAT3HTT
Triaziquone SCHEMBL10414999 0.83 MAPT (0.41) DNMT1MAPTTP53STAT3HTT
Triaziquone SCHEMBL8926769 0.83 DNMT1 (0.42) DNMT1MAPTTP53STAT3HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006079364-A1 SPECIFIC AND MILD PEPTIDE OR AMIDE BOND CLEAVAGE STICHTING VOOR DE TECHNISCHE WETENSCHAPPEN (NL) 2006-08-03 WO claimed
CN-115023610-A Novel linker compounds 剑桥实业有限公司 2022-09-06 CN disclosed
EP-2084295-A2 METHOD FOR SEQUENCING A POLYNUCLEOTIDE TEMPLATE Illumina Cambridge Limited (GB) 2009-08-05 EP disclosed
EP-1987159-A1 METHOD FOR SEQUENCING A POLYNUCLEOTIDE TEMPLATE Illumina Cambridge Limited (GB) 2008-11-05 EP disclosed
EP-1910561-A1 METHODS OF NUCLEIC ACID AMPLIFICATION AND SEQUENCING Solexa Ltd. (GB) 2008-04-16 EP disclosed
EP-1910560-A1 METHOD FOR SEQUENCING A POLYNUCLEOTIDE TEMPLATE Solexa Ltd. (GB) 2008-04-16 EP disclosed
EP-1910559-A2 PREPARATION OF TEMPLATES FOR NUCLEIC ACID SEQUENCING Solexa Ltd. (GB) 2008-04-16 EP disclosed
WO-2008041002-A2 METHOD FOR SEQUENCING A POLYNUCLEOTIDE TEMPLATE ILLUMINA CAMBRIDGE LIMITED (GB) 2008-04-10 WO disclosed
EP-1799846-A4 METHODS FOR ISOLATING NUCLEIC ACIDS FROM BIOLOGICAL AND CELLULAR MATERIALS NEXGEN DIAGNOSTICS LLC (US) 2008-01-16 EP disclosed
EP-1828412-A1 IMPROVED METHOD OF NUCLEOTIDE DETECTION Solexa Ltd. (GB) 2007-09-05 EP disclosed
WO-2007091077-A1 METHOD FOR SEQUENCING A POLYNUCLEOTIDE TEMPLATE SOLEXA LIMITED (GB) 2007-08-16 WO disclosed
EP-1799846-A2 METHODS FOR ISOLATING NUCLEIC ACIDS FROM BIOLOGICAL AND CELLULAR MATERIALS LUMIGEN, INC. (US) 2007-06-27 EP disclosed
WO-2007010251-A2 PREPARATION OF TEMPLATES FOR NUCLEIC ACID SEQUENCING SOLEXA LIMITED (GB) 2007-01-25 WO disclosed
WO-2007010252-A1 METHOD FOR SEQUENCING A POLYNUCLEOTIDE TEMPLATE SOLEXA LIMITED (GB) 2007-01-25 WO disclosed
WO-2007010254-A1 METHODS OF NUCLEIC ACID AMPLIFICATION AND SEQUENCING SOLEXA LIMITED (GB) 2007-01-25 WO disclosed
WO-2006079364-A1 SPECIFIC AND MILD PEPTIDE OR AMIDE BOND CLEAVAGE STICHTING VOOR DE TECHNISCHE WETENSCHAPPEN (NL) 2006-08-03 WO disclosed
WO-2006064199-A1 IMPROVED METHOD OF NUCLEOTIDE DETECTION SOLEXA LIMITED (GB) 2006-06-22 WO disclosed
WO-2006036243-A2 METHODS FOR ISOLATING NUCLEIC ACIDS FROM BIOLOGICAL AND CELLULAR MATERIALS LUMIGEN, INC. (US) 2006-04-06 WO disclosed