SCHEMBL4084332

SCHEMBL4084332

CN(C)C1(c2cccs2)CCC(NC(=O)CCC(=O)N2CCC(O)(c3ccc(C(F)(F)F)cc3)CC2)CC1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 3/20 0.43
OPRL1 P41146 3/20 0.43
EPHX2 P34913 4/20 0.41
CCR2 P41597 5/20 0.40
KCNH2 Q12809 4/20 0.40
DRD2 P14416 2/20 0.38
ENPP2 Q13822 1/20 0.38
DRD4 P21917 1/20 0.38
DRD3 P35462 1/20 0.38
S1PR2 O95136 1/20 0.37
KMT2A Q03164 1/20 0.37
CCRL2 O00421 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL208749 0.92 CCR2 (0.45) OPRM1OPRL1CCR2KCNH2
SCHEMBL207647 0.83 KDM4E (0.46) KMT2A
SCHEMBL206307 0.81 OPRM1 (0.52) OPRM1OPRL1CCR2KCNH2
SCHEMBL5158003 0.79 CHRM4 (0.42) OPRM1OPRL1CCR2KCNH2
SCHEMBL206822 0.78 OPRM1 (0.47) OPRM1OPRL1KMT2A
SCHEMBL206118 0.77 HDAC3 (0.45) OPRM1OPRL1CCR2KCNH2
SCHEMBL206198 0.76 ALDH1A1 (0.45) KMT2A
SCHEMBL4074077 0.76 OPRM1 (0.51) OPRM1OPRL1EPHX2
SCHEMBL206119 0.75 OPRM1 (0.43) OPRM1OPRL1CCR2KCNH2DRD2
SCHEMBL208760 0.74 SMYD3 (0.48) OPRM1OPRL1CCR2KCNH2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1745010-B1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES GRUENENTHAL GMBH (DE) 2009-08-05 EP claimed