SCHEMBL4085714

SCHEMBL4085714

CCCCc1c(-c2ccc(-c3nc(Nc4ccc(Cn5ccnc5C)cc4)nc4[nH]ccc34)s2)cccc1S(N)(=O)=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK1 P23458 2/20 0.38
JAK2 O60674 6/20 0.33
HDAC1 Q13547 2/20 0.33
HDAC6 Q9UBN7 2/20 0.33
CDK1 P06493 4/20 0.33
CDK5 Q00535 4/20 0.33
CDK2 P24941 2/20 0.33
CCNT1 O60563 1/20 0.33
CCNB1 P14635 1/20 0.33
CDK7 P50613 1/20 0.33
CDK9 P50750 1/20 0.33
CCNH P51946 1/20 0.33
AGTR2 P50052 2/20 0.32
KDR P35968 5/20 0.32
CA1 P00915 2/20 0.32
CA2 P00918 2/20 0.32
CA9 Q16790 2/20 0.32
TNIK Q9UKE5 1/20 0.32
CA12 O43570 1/20 0.32
AURKA O14965 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13883626 0.83 IKBKB (0.41) JAK1JAK2CDK1CDK5CDK2
SCHEMBL4085715 0.80 JAK1 (0.39) JAK1JAK2HDAC1HDAC6CDK5
SCHEMBL13883576 0.78 JAK2 (0.40) JAK1JAK2CDK5KDRTNIK
SCHEMBL4407227 0.78 JAK1 (0.38) JAK1JAK2HDAC1CDK7CDK9
SCHEMBL13883718 0.77 AXL (0.38) JAK1JAK2TNIKPDPK1
SCHEMBL4255795 0.76 JAK1 (0.38) JAK1JAK2HDAC1HDAC6CDK5
SCHEMBL4409833 0.74 TNIK (0.37) JAK1JAK2HDAC1HDAC6CDK5
SCHEMBL3971650 0.74 TNIK (0.39) JAK1JAK2HDAC1HDAC6AGTR2
SCHEMBL3973621 0.74 JAK2 (0.38) JAK1JAK2CDK5KDRTNIK
SCHEMBL4081315 0.74 AXL (0.46) JAK2CDK1KDRAURKAJAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009049028-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USE AS JANUS KINASE MODULATORS TARGEGEN INC. (US) 2009-04-16 WO claimed