SCHEMBL4086659

SCHEMBL4086659

CC(C)(C)[S+]([O-])NCc1ccc2cccnc2c1-c1cc(F)cc(F)c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 1/20 0.34
SLC40A1 Q9NP59 2/20 0.34
CKS1B P61024 1/20 0.33
SKP2 Q13309 1/20 0.33
EGLN1 Q9GZT9 1/20 0.32
MAPT P10636 3/20 0.32
KDM4E B2RXH2 2/20 0.32
CCR1 P32246 2/20 0.32
CCR5 P51681 2/20 0.32
CCR8 P51685 2/20 0.32
LMNA P02545 2/20 0.32
MMP2 P08253 2/20 0.32
TP53 P04637 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
GMNN O75496 1/20 0.32
HSP90AA1 P07900 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
MMP9 P14780 1/20 0.32
ALOX15 P16050 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2721580 0.89 PIK3CD (0.33) PIK3CDSLC40A1CKS1BSKP2MAPT
SCHEMBL2721578 0.77 PIK3CD (0.45) PIK3CDSLC40A1CKS1BSKP2MAPT
SCHEMBL2718191 0.75 KDM4E (0.42) EGLN1MAPTKDM4ECCR1CCR5
SCHEMBL2011511 0.73 KDM4E (0.40) EGLN1MAPTKDM4ECCR1CCR5
SCHEMBL2011836 0.73 LMNA (0.40) SLC40A1MAPTKDM4ECCR1CCR5
SCHEMBL2016022 0.72 CCR1 (0.39) SLC40A1CKS1BSKP2EGLN1MAPT
SCHEMBL2719983 0.72 MET (0.34) PIK3CDSLC40A1CKS1BSKP2MAPT
SCHEMBL2719987 0.72 MET (0.34) PIK3CDSLC40A1CKS1BSKP2MAPT
SCHEMBL2718705 0.71 HPGD (0.32) TDP1
SCHEMBL4078039 0.67 PTGDR2 (0.37) MAPTMMP2MMP9MMP13MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012061696-A1 5 -CYANO-4, 6 -DIAMINOPYRIMIDINE OR 6 -AMINOPURINE DERIVATIVES AS PI3K- DELTA INHIBITORS AMGEN INC. (US) 2012-05-10 WO disclosed