SCHEMBL4092903

SCHEMBL4092903

CC(C)(NC(=O)c1cc2[nH]nc(NC(=O)c3ccc(CN4CCCC4)cc3)c2o1)c1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 2/20 0.61
BCR P11274 2/20 0.61
AURKA O14965 3/20 0.50
HRH3 Q9Y5N1 2/20 0.44
ACKR3 P25106 1/20 0.44
CYP2C9 P11712 1/20 0.44
HIF1A Q16665 2/20 0.43
EPAS1 Q99814 2/20 0.43
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPT P10636 1/20 0.42
RAB9A P51151 1/20 0.42
KIT P10721 2/20 0.42
FLT3 P36888 1/20 0.42
KDR P35968 2/20 0.41
HDAC1 Q13547 3/20 0.40
HDAC4 P56524 1/20 0.40
KCNH2 Q12809 1/20 0.40
CDC7 O00311 1/20 0.40
CHEK1 O14757 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4093502 0.99 ABL1 (0.63) ABL1BCRAURKAHRH3ACKR3
SCHEMBL4083868 0.98 ABL1 (0.59) ABL1BCRAURKAHRH3ACKR3
SCHEMBL4081436 0.94 AURKA (0.57) ABL1BCRAURKAACKR3HIF1A
SCHEMBL4081465 0.94 ABL1 (0.54) ABL1BCRAURKAHIF1AEPAS1
SCHEMBL4088412 0.90 ABL1 (0.51) ABL1BCRAURKAHRH3CYP2C9
SCHEMBL4086294 0.89 ABL1 (0.52) ABL1BCRAURKAHRH3CYP2C9
SCHEMBL4082984 0.87 AURKA (0.48) ABL1BCRAURKAKITFLT3
SCHEMBL4088217 0.87 AURKA (0.51) ABL1BCRAURKAJAK2FGFR1
SCHEMBL4092679 0.86 AURKA (0.49) ABL1BCRAURKAACKR3KDM4E
SCHEMBL4082914 0.85 HRH3 (0.48) ABL1BCRAURKAHRH3CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2058315-A1 1H-Furo[3,2-C]Pyrazoles active as aurora kinase inhibitors Nerviano Medical Sciences S.r.l. (IT) 2009-05-13 EP disclosed