SCHEMBL4095238

SCHEMBL4095238

CC(C)n1cc(C(=O)CC#N)c2cccc(Br)c21

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.35
ALDH1A1 P00352 4/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
HK1 P19367 1/20 0.35
HKDC1 Q2TB90 1/20 0.35
KDM4E B2RXH2 1/20 0.34
HTT P42858 3/20 0.33
LMNA P02545 2/20 0.33
TSHR P16473 3/20 0.33
CNR1 P21554 1/20 0.32
CNR2 P34972 1/20 0.32
MAPT P10636 3/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C19 P33261 1/20 0.32
HSP90AA1 P07900 1/20 0.32
HPGD P15428 1/20 0.32
FGFR4 P22455 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4095742 0.80 BRD4 (0.40) ALDH1A1SMN1; SMN2KDM4EHTTLMNA
SCHEMBL4084945 0.76 DYRK1A (0.41) ALDH1A1SMN1; SMN2KDM4E
SCHEMBL13885188 0.71 JAK3 (0.38) KCNH2
SCHEMBL30605772 0.68 MAPT (0.49) KCNH2ALDH1A1SMN1; SMN2KDM4EHTT
SCHEMBL1998027 0.68 MAPT (0.49) KCNH2ALDH1A1SMN1; SMN2KDM4EHTT
SCHEMBL2599810 0.68 ALDH1A1 (0.40) ALDH1A1SMN1; SMN2KDM4EHTTLMNA
SCHEMBL4094763 0.68 PDE4B (0.32) ALDH1A1CYP1A2
SCHEMBL5676525 0.66 KCNH2 (0.43) KCNH2ALDH1A1SMN1; SMN2HK1HKDC1
SCHEMBL20838602 0.66 ALDH1A1 (0.66) ALDH1A1SMN1; SMN2HK1HKDC1KDM4E
SCHEMBL29426296 0.66 ALDH1A1 (0.66) ALDH1A1SMN1; SMN2HK1HKDC1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009055674-A1 PYRROLOPYRIMIDINE ALKYNYL COMPOUNDS AND METHODS OF MAKING AND USING SAME TARGEGEN INC. (US) 2009-04-30 WO disclosed
WO-2009055674-A1 PYRROLOPYRIMIDINE ALKYNYL COMPOUNDS AND METHODS OF MAKING AND USING SAME TARGEGEN INC. (US) 2009-04-30 WO disclosed