SCHEMBL4100978

SCHEMBL4100978

COc1ccc(Cn2cc(C)c(-c3ccco3)c2OC(=O)O)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.43
CHRM1 P11229 1/20 0.42
ADORA2A P29274 1/20 0.42
SIRT1 Q96EB6 1/20 0.40
MAPT P10636 3/20 0.40
THRB P10828 1/20 0.40
LMNA P02545 3/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
POLB P06746 1/20 0.39
MAPK1 P28482 2/20 0.39
UBE2I P63279 1/20 0.39
CACNA1B Q00975 1/20 0.39
APBA1 Q02410 1/20 0.39
SAE1 Q9UBE0 1/20 0.39
UBA2 Q9UBT2 1/20 0.39
KMT2A Q03164 3/20 0.38
RAB9A P51151 1/20 0.38
TSHR P16473 2/20 0.38
HSD17B10 Q99714 2/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4122565 0.88 ALDH1A1 (0.41) ALDH1A1SMN1; SMN2POLBMAPK1KMT2A
SCHEMBL1032311 0.85 ADORA2A (0.41) ALDH1A1ADORA2ALMNASMN1; SMN2POLB
SCHEMBL2637910 0.85 TP53 (0.44) ALDH1A1CHRM1ADORA2ASIRT1MAPT
SCHEMBL4102629 0.80 LMNA (0.44) ALDH1A1CHRM1LMNASMN1; SMN2POLB
SCHEMBL4109233 0.78 SMN1; SMN2 (0.45) ALDH1A1CHRM1MAPTTHRBLMNA
SCHEMBL1032103 0.77 TAS1R3 (0.43) ALDH1A1POLBUBE2ICACNA1BAPBA1
SCHEMBL1027735 0.76 ALDH1A1 (0.53) ALDH1A1MAPTLMNAPOLBKMT2A
SCHEMBL1030275 0.75 L3MBTL1 (0.40) ALDH1A1MAPTTHRBLMNAPOLB
SCHEMBL1030586 0.75 ALDH1A1 (0.41) ALDH1A1ADORA2AMAPTTHRBPOLB
SCHEMBL1031303 0.74 GAA (0.42) ALDH1A1MAPTLMNAPOLBMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2035375-A1 1,3-DISUBSTITUTED 4-METHYL-1H-PYRROLE-2-CARBOXAMIDES AND THEIR USE FOR THE MANUFACTURE OF MEDICAMENTS Grünenthal GmbH (DE) 2009-03-18 EP claimed
WO-2007141039-A1 1,3-DISUBSTITUTED 4-METHYL-1H-PYRROLE-2-CARBOXAMIDES AND THEIR USE FOR THE MANUFACTURE OF MEDICAMENTS Grünenthal GmbH (DE) 2007-12-13 WO claimed
EP-2035375-A1 1,3-DISUBSTITUTED 4-METHYL-1H-PYRROLE-2-CARBOXAMIDES AND THEIR USE FOR THE MANUFACTURE OF MEDICAMENTS Grünenthal GmbH (DE) 2009-03-18 EP disclosed
WO-2007141039-A1 1,3-DISUBSTITUTED 4-METHYL-1H-PYRROLE-2-CARBOXAMIDES AND THEIR USE FOR THE MANUFACTURE OF MEDICAMENTS Grünenthal GmbH (DE) 2007-12-13 WO disclosed