Benzamil

Benzamil

SCHEMBL412783

N/C(=N\C(=O)c1nc(Cl)c(N)nc1N)NCc1ccccc1

nearest known ligand 0.63

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLAU P00749 9/20 0.63
SCNN1A P37088 9/20 0.58
ALDH1A1 P00352 6/20 0.58
KDM4E B2RXH2 5/20 0.58
GLA P06280 5/20 0.58
HPGD P15428 5/20 0.58
HSD17B10 Q99714 5/20 0.58
GAA P10253 3/20 0.58
CYP1A2 P05177 3/20 0.58
CYP2D6 P10635 2/20 0.58
FTO Q9C0B1 2/20 0.58
TDP1 Q9NUW8 2/20 0.58
NPC1 O15118 2/20 0.58
MAPT P10636 1/20 0.58
NFKB1 P19838 1/20 0.58
THPO P40225 1/20 0.58
HIF1A Q16665 1/20 0.58
BLM P54132 2/20 0.57
GMNN O75496 1/20 0.57
PMP22 Q01453 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Benzamil SCHEMBL5433990 1.00 PLAU (0.63) PLAUSCNN1AALDH1A1KDM4EGLA
Benzamil SCHEMBL4242779 1.00 PLAU (0.63) PLAUSCNN1AALDH1A1KDM4EGLA
Benzamil SCHEMBL9464171 0.99 PLAU (0.64) PLAUSCNN1AALDH1A1KDM4EGLA
SCHEMBL11615365 0.94 PLAU (0.59) PLAUSCNN1AALDH1A1KDM4EGLA
SCHEMBL10028719 0.85 SCNN1A (0.61) PLAUSCNN1AALDH1A1KDM4EGLA
3',4' Dichlorobenzamil SCHEMBL14504158 0.85 HSD17B10 (0.60) PLAUSCNN1AALDH1A1KDM4EGLA
SCHEMBL5065784 0.83 KCNH2 (0.51) PLAUSCNN1AALDH1A1KDM4EGLA
SCHEMBL5014171 0.82 SCNN1A (0.52) PLAUSCNN1AALDH1A1KDM4EGLA
Phenamil SCHEMBL14504131 0.81 PLAU (0.58) PLAUSCNN1AALDH1A1KDM4EGLA
Phenamil SCHEMBL14973571 0.81 PLAU (0.58) PLAUSCNN1AALDH1A1KDM4EGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1958 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250057876-A1 METHODS FOR TREATING AND/OR PREVENTING LYMPHANGIOGENESIS-ASSOCIATED DISEASES BY USING GOLD NANOCLUSTERS GOLDRED NANOBIOTECH CO., LTD. (TW) 2025-02-20 US claimed
US-20250009739-A1 METHOD OF TREATING A SKIN DISORDER PHAMRI NORDEN AB (SE) 2025-01-09 US claimed
US-20250002463-A1 NEW SALT FORMS OF AMILORIDE AND ITS DERIVATIVES FOR PHARMACEUTICAL USE PSOMRI HOLDING AB (SE) 2025-01-02 US claimed
EP-4408826-A1 NEW SALT FORMS OF AMILORIDE AND ITS DERIVATIVES FOR PHARMACEUTICAL USE Psomri Holding AB (SE) 2024-08-07 EP claimed
US-20240180955-A1 FIBER SUPPLEMENTATION PROTECTS FROM ANTIBIOTIC-INDUCED GUT MICROBIOME DYSBIOSIS BY MODULATING REDOX METABOLISM BROWN UNIVERSITY 2024-06-06 US claimed
EP-4281075-A2 METHOD OF TREATING A SKIN DISORDER BY ADMINISTERING AN AMILORIDE DERIVATIVE Pharmi Norden AB (SE) 2023-11-29 EP claimed
US-11826366-B2 Composition and methods for preventing or reducing the incidence of transient ischemic attacks MOREHOUSE SCHOOL OF MEDICINE (US) 2023-11-28 US claimed
US-11819535-B2 Composition and methods for regulating extracellular matrix accumulation UNIVERSITY HEALTH NETWORK (CA) 2023-11-21 US claimed
WO-2023183932-A2 MONOBODIES BINDING TO INTERCELLULAR ADHESION MOLECULE 2 (ICAM-2) NEW YORK UNIVERSITY (US) 2023-09-28 WO claimed
WO-2023066893-A1 AMILORIDE DERIVATIVES FOR TREATING INFLAMMATION IN THE INTESTINES PHAMRI NORDEN AB (SE) 2023-04-27 WO claimed
EP-0778768-A1 FORMULATIONS AND METHODS FOR PROVIDING PROLONGED LOCAL ANESTHESIA Euroceltique S.A. (LU) 1997-06-18 EP claimed
US-5635160-A Dinucleotides useful for the treatment of cystic fibrosis and for hydrating mucus secretions THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 1997-06-03 US claimed
US-5628984-A Method of detecting lung disease UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 1997-05-13 US claimed
WO-1997005195-A1 METHOD OF DETECTING LUNG DISEASE THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 1997-02-13 WO claimed
WO-1996041616-A1 FORMULATIONS AND METHODS FOR PROVIDING PROLONGED LOCAL ANESTHESIA EURO-CELTIQUE, S.A. (LU) 1996-12-27 WO claimed
WO-1996040059-A1 DINUCLEOTIDES USEFUL FOR THE TREATMENT OF LUNG DISEASE THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 1996-12-19 WO claimed
WO-1996018385-A1 METHODS OF TREATING LUNG DISEASE THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 1996-06-20 WO claimed
WO-1996013158-A2 PROLONGED PRESERVATION OF BLOOD PLATELETS LIFECELL CORPORATION (US) 1996-05-09 WO claimed
EP-0451130-A2 Use of amiloride and other pyrazine derivatives for preventing or treating ocular neovascularization CELTRIX PHARMACEUTICALS, INC. (US) 1991-10-09 EP claimed
US-4894376-A Methods of treating diseases characterized by hyperexcitability of neurons TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 1990-01-16 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250009739-A1 METHOD OF TREATING A SKIN DISORDER CUTA, KRT18, ASAH2 PLAU 216/4885SCNN1A 255/4885ALDH1A1 345/4885
US-20250002463-A1 NEW SALT FORMS OF AMILORIDE AND ITS DERIVATIVES FOR PHARMACEUTICAL USE ASIC1, PPA1, ASIC3 PLAU 1690/4885SCNN1A 175/4885ALDH1A1 428/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.