SCHEMBL4131797

SCHEMBL4131797

O=C(NNC(=S)NCCCCN1CCCC1)c1c[nH]c2ccccc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.56
DRD3 P35462 2/20 0.54
HTR1A P08908 1/20 0.54
HTR2A P28223 1/20 0.54
HTR2C P28335 1/20 0.54
KMT2A Q03164 1/20 0.53
HTR4 Q13639 2/20 0.51
ALDH1A1 P00352 1/20 0.51
CYP1A2 P05177 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
TSHR P16473 1/20 0.51
THPO P40225 1/20 0.51
PMP22 Q01453 1/20 0.50
HRH3 Q9Y5N1 1/20 0.50
HDAC1 Q13547 2/20 0.48
HDAC2 Q92769 2/20 0.48
HDAC3 O15379 1/20 0.48
HDAC4 P56524 1/20 0.48
HDAC7 Q8WUI4 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7330236 0.79 KMT2A (0.67) DRD2DRD3HTR1AHTR2AHTR2C
SCHEMBL3999744 0.79 CCR2 (0.47) KMT2AALDH1A1CCR2
SCHEMBL4131795 0.77 ALDH1A1 (0.50) DRD2DRD3HTR1AHTR2AHTR2C
SCHEMBL9661528 0.75 DRD2 (0.62) DRD2DRD3HTR1AHTR2AHTR2C
SCHEMBL3997685 0.73 HDAC1 (0.50) ALDH1A1CYP1A2CYP2D6TSHRHDAC1
SCHEMBL4245219 0.72 HTR3A (0.57) KMT2AALDH1A1
SCHEMBL9650947 0.72 DRD3 (0.75) DRD2DRD3HTR1AHTR2AHTR2C
SCHEMBL4003759 0.72 SMYD2 (0.47)
SCHEMBL24651274 0.72 NR1I2 (0.63) DRD2DRD3HTR1AHTR2AHTR2C
SCHEMBL9661440 0.71 DRD2 (0.58) DRD2DRD3HTR1AHTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009071577-A1 OXADIAZOLE DERIVATIVES AND THEIR USE AS NICOTINIC ACETYLCHOLINE RECEPTOR MODULATORS GLAXO GROUP LIMITED (GB) 2009-06-11 WO disclosed
WO-2009071577-A1 OXADIAZOLE DERIVATIVES AND THEIR USE AS NICOTINIC ACETYLCHOLINE RECEPTOR MODULATORS GLAXO GROUP LIMITED (GB) 2009-06-11 WO disclosed