SCHEMBL4132982

SCHEMBL4132982

C[SiH](C)OC(c1c(OCc2ccc(C#N)nc2)ccc2c(CCC3CCN(C(=O)OC(C)(C)C)CC3)noc12)C(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 12/20 0.38
CETP P11597 2/20 0.34
JAK2 O60674 1/20 0.34
JAK1 P23458 1/20 0.34
YAP1 P46937 2/20 0.34
NSD2 O96028 1/20 0.33
EHMT2 Q96KQ7 1/20 0.33
CSF1R P07333 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4126342 0.93 ACHE (0.35) JAK2JAK1
SCHEMBL4119097 0.88 GPR119 (0.37) GPR119YAP1
SCHEMBL4126973 0.88 HTT (0.38) GPR119YAP1
SCHEMBL4122093 0.87 CETP (0.37) GPR119CETPNSD2
SCHEMBL4132983 0.83 GPR119 (0.40) GPR119JAK2JAK1YAP1CSF1R
SCHEMBL4122090 0.82 FAAH (0.37) GPR119CETPCSF1R
SCHEMBL4120553 0.81 GPR119 (0.38) GPR119CETPCSF1R
SCHEMBL4127266 0.80 ACHE (0.39) YAP1
SCHEMBL4124936 0.80 HTT (0.39)
SCHEMBL4127069 0.80 GPR119 (0.36) GPR119CETP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090318690-A1 Benzisoxazole Compound EISAI R&D MANAGEMENT CO., LTD. (JP) 2009-12-24 US disclosed
EP-2017275-A1 BENZISOXAZOLE COMPOUND Eisai R&D Management Co., Ltd. (JP) 2009-01-21 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090318690-A1 Benzisoxazole Compound NR1I2, NR1I3, NR0B1 GPR119 122/4885CETP 3157/4885JAK2 1131/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.