SCHEMBL4135822

SCHEMBL4135822

COc1cc(CC=O)ccc1N1CCC2(CC1)CCN(C1CCC1)CC2

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.45
ALDH1A3 P47895 1/20 0.45
FFAR4 Q5NUL3 5/20 0.41
DRD2 P14416 2/20 0.39
MAPT P10636 1/20 0.38
DRD3 P35462 1/20 0.38
FLT3 P36888 1/20 0.37
HTR1A P08908 1/20 0.37
ADRA1D P25100 1/20 0.37
ADRA1A P35348 1/20 0.37
ADRA1B P35368 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
POLB P06746 1/20 0.36
SIGMAR1 Q99720 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4130771 0.83 ALDH1A1 (0.42) ALDH1A1FFAR4
SCHEMBL4135820 0.79 ALDH1A1 (0.44) ALDH1A1ALDH1A3FFAR4
SCHEMBL4136516 0.79 HRH3 (0.47) FFAR4
SCHEMBL4123180 0.76 HRH3 (0.39) ALDH1A1FFAR4MEN1KMT2A
SCHEMBL4141352 0.76 FFAR4 (0.48) ALDH1A1FFAR4
SCHEMBL4135581 0.72 TLR9 (0.38) FFAR4ADRA1APOLB
SCHEMBL16440170 0.70 ALDH1A1 (0.56) ALDH1A1ALDH1A3DRD2HTR1AADRA1D
SCHEMBL4140025 0.70 SCD (0.40) MAPTMEN1KMT2A
SCHEMBL4135176 0.68 HRH3 (0.38) FFAR4
SCHEMBL4146899 0.68 KDM2B (0.45) ALDH1A1FFAR4MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2021004-A2 SUBSTITUTED AZASPIRO DERIVATIVES NEUROGEN CORPORATION (US) 2009-02-11 EP claimed
WO-2007133561-A2 SUBSTITUTED AZASPIRO DERIVATIVES NEUROGEN CORPORATION (US) 2007-11-22 WO claimed