SCHEMBL413751

SCHEMBL413751

COC(=O)c1ccc(NCC2=CC(=O)c3ccccc3C2=O)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 1.00
CA1 P00915 4/20 0.57
CA2 P00918 4/20 0.57
CDC25B P30305 3/20 0.55
PTPRC P08575 1/20 0.55
PTPRF P10586 1/20 0.55
PTPN1 P18031 1/20 0.55
CDC25A P30304 2/20 0.51
SMN1; SMN2 Q16637 3/20 0.49
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
HPGD P15428 2/20 0.49
MAPT P10636 2/20 0.49
HTT P42858 2/20 0.49
HKDC1 Q2TB90 2/20 0.49
KDM4E B2RXH2 1/20 0.49
APAF1 O14727 1/20 0.49
MITF O75030 1/20 0.49
THRB P10828 1/20 0.49
NR4A1 P22736 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL413750 0.78 CYP19A1 (0.63) CYP19A1CDC25BPTPN1CDC25ASMN1; SMN2
SCHEMBL30704429 0.77 RAB9A (0.67) CYP19A1CDC25BPTPRCPTPRFPTPN1
SCHEMBL15690558 0.77 CYP19A1 (0.62) CYP19A1CA1CA2CDC25BPTPRC
SCHEMBL412798 0.76 CYP19A1 (0.61) CYP19A1CA1CA2SMN1; SMN2MEN1
SCHEMBL16938319 0.74 CYP19A1 (0.59) CYP19A1CA1CA2CDC25BPTPRC
SCHEMBL18415526 0.73 CA1 (1.00) CYP19A1CA1CA2SMN1; SMN2MEN1
SCHEMBL30704447 0.72 GAPDH (0.63) CYP19A1CA1CA2CDC25BPTPRC
SCHEMBL11412192 0.72 CYP19A1 (0.56) CYP19A1CDC25BPTPRCPTPRFPTPN1
SCHEMBL15514574 0.71 CDC25B (0.55) CYP19A1CDC25BPTPRCPTPRFPTPN1
SCHEMBL13934091 0.71 CA1 (0.87) CYP19A1CA1CA2SMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120021519-A1 EFFICIENT INDUCTION OF PLURIPOTENT STEM CELLS USING SMALL MOLECULE COMPOUNDS PRESIDENTS AND FELLOWS OF HARVARD COLLEGE (US) 2012-01-26 US disclosed
WO-2010033906-A2 EFFICIENT INDUCTION OF PLURIPOTENT STEM CELLS USING SMALL MOLECULE COMPOUNDS PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2010-03-25 WO disclosed