SCHEMBL4138734

SCHEMBL4138734

Fc1c(F)c(F)c(-c2ccc(C(F)(F)F)cc2)c(F)c1F

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 9/20 0.52
ALDH1A1 P00352 1/20 0.42
TSHR P16473 1/20 0.42
MAOB P27338 1/20 0.41
HEXA P06865 1/20 0.40
HEXB P07686 1/20 0.40
BACE1 P56817 1/20 0.39
CES2 O00748 1/20 0.39
CES1 P23141 1/20 0.39
ORAI1 Q96D31 1/20 0.39
ORAI2 Q96SN7 1/20 0.39
ORAI3 Q9BRQ5 1/20 0.39
TRPV6 Q9H1D0 1/20 0.39
MGLL Q99685 1/20 0.39
NISCH Q9Y2I1 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21001760 0.86 KIF11 (0.48) KIF11ALDH1A1TSHRMAOBHEXA
SCHEMBL31409757 0.86 KIF11 (0.48) KIF11ALDH1A1TSHRMAOBHEXA
SCHEMBL28248236 0.84 KIF11 (0.46) KIF11ALDH1A1TSHRMAOB
SCHEMBL20769886 0.82 KIF11 (0.48) KIF11HEXAHEXBNISCH
SCHEMBL17711075 0.82 KIF11 (0.53) KIF11ALDH1A1
SCHEMBL4159679 0.81 TTR (0.32)
SCHEMBL27256051 0.80 KIF11 (0.53) KIF11ALDH1A1TSHRBACE1TRPV6
SCHEMBL12762364 0.78 KIF11 (0.46) KIF11ALDH1A1TSHRMAOBNISCH
SCHEMBL197238 0.78 KIF11 (0.78) KIF11ALDH1A1TSHRMAOBCES2
SCHEMBL29914837 0.78 KIF11 (0.78) KIF11ALDH1A1TSHRMAOBCES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113429259-B Fluorine-containing compound and application thereof 中国科学院上海有机化学研究所 2023-03-24 CN disclosed
US-8952207-B2 Copper-catalyzed C—H bond arylation THE UNIVERSITY OF HOUSTON SYSTEM (US) 2015-02-10 US disclosed
US-8952207-B2 Copper-catalyzed C—H bond arylation THE UNIVERSITY OF HOUSTON SYSTEM (US) 2015-02-10 US disclosed
US-8952207-B2 Copper-catalyzed C—H bond arylation THE UNIVERSITY OF HOUSTON SYSTEM (US) 2015-02-10 US disclosed
US-20090076266-A1 COPPER-CATALYZED C-H BOND ARYLATION THE UNIVERSITY OF HOUSTON SYSTEM (US) 2009-03-19 US disclosed
US-20090076266-A1 COPPER-CATALYZED C-H BOND ARYLATION THE UNIVERSITY OF HOUSTON SYSTEM (US) 2009-03-19 US disclosed
US-20090076266-A1 COPPER-CATALYZED C-H BOND ARYLATION THE UNIVERSITY OF HOUSTON SYSTEM (US) 2009-03-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090076266-A1 COPPER-CATALYZED C-H BOND ARYLATION AOC2, AOC3, DBH KIF11 1251/4885ALDH1A1 44/4885TSHR 3189/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.