SCHEMBL4145160

SCHEMBL4145160

CCOCN(C(=O)Nc1ccc(SC(F)(F)F)cc1F)C(=O)c1c(F)cccc1F

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
RXFP1 Q9HBX9 2/20 0.37
HTT P42858 2/20 0.34
PPARG P37231 1/20 0.34
PPARD Q03181 1/20 0.34
PPARA Q07869 1/20 0.34
BRAF P15056 1/20 0.34
MAPT P10636 1/20 0.33
HDAC4 P56524 1/20 0.33
MEF2D Q14814 1/20 0.33
KCNK2 O95069 4/20 0.32
TRPA1 O75762 2/20 0.32
TRPV1 Q8NER1 1/20 0.32
CYP1A2 P05177 1/20 0.32
DHODH Q02127 2/20 0.32
KCNK10 P57789 2/20 0.31
PKM P14618 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4149970 0.90 RXFP1 (0.35) RXFP1HTTBRAFKCNK2TRPA1
SCHEMBL4636108 0.90 RXFP1 (0.39) RXFP1HTTPPARGPPARDPPARA
SCHEMBL4150571 0.89 BRAF (0.33) RXFP1HTTBRAFKCNK2KCNK10
SCHEMBL5311662 0.88 BRAF (0.33) RXFP1HTTPPARGPPARDPPARA
SCHEMBL4141961 0.88 PPARG (0.37) RXFP1PPARGPPARDPPARABRAF
SCHEMBL5313986 0.85 HTT (0.36) RXFP1HTTPPARGPPARDPPARA
SCHEMBL5335591 0.82 HTT (0.34) HTTPPARGPPARDPPARAMAPT
SCHEMBL5314985 0.82 HTT (0.43) RXFP1HTTPPARGPPARDPPARA
SCHEMBL5316114 0.82 KMT2A (0.35) RXFP1HTTBRAFMAPTKCNK2
SCHEMBL5316133 0.82 POLB (0.39) RXFP1MAPTKCNK2DHODHKCNK10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090176786-A1 Benzoylurea Compounds and Use Thereof SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2009-07-09 US disclosed
US-20090176786-A1 Benzoylurea Compounds and Use Thereof SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2009-07-09 US disclosed
EP-1937629-A2 BENZOYLUREA COMPOUNDS AND USE THEREOF Sumitomo Chemical Company, Limited (JP) 2008-07-02 EP disclosed
WO-2007066496-A1 BENZOYLUREA COMPOUND AND USE THEREOF SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2007-06-14 WO disclosed
WO-2007046513-A2 BENZOYLUREA COMPOUNDS AND USE THEREOF SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2007-04-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090176786-A1 Benzoylurea Compounds and Use Thereof BTK, BRIX1, NFXL1 RXFP1 832/4885HTT 2562/4885PPARG 3528/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.