SCHEMBL4147

SCHEMBL4147

Cc1noc(-c2ccc(-c3ccc(C4(CC(=O)O)CC4)cc3)cc2)c1N(C)CCc1ccc(OCc2ccc(C(F)(F)F)cc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PPARD Q03181 9/20 0.43
PPARG P37231 7/20 0.43
PPARA Q07869 6/20 0.43
FFAR1 O14842 7/20 0.42
SMPD1 P17405 1/20 0.39
PTGDR2 Q9Y5Y4 2/20 0.39
FFAR4 Q5NUL3 1/20 0.37
MAOB P27338 1/20 0.37
ADAMTS4 O75173 1/20 0.36
MMP13 P45452 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7026 0.86 AOC3 (0.37) FFAR4
SCHEMBL6613 0.81 FFAR4 (0.35) FFAR4
SCHEMBL14854 0.81 PPARD (0.42) PPARDPPARGPPARAFFAR1SMPD1
SCHEMBL6082 0.79 HDAC1 (0.34) PPARDPPARGPPARAFFAR4
SCHEMBL7148 0.78 ALDH1A1 (0.38) FFAR1FFAR4
SCHEMBL6973 0.77 BRD4 (0.36)
SCHEMBL7534 0.75 L3MBTL1 (0.34)
SCHEMBL7666 0.74 ABCC3 (0.44)
SCHEMBL7297 0.73 SCD5 (0.35)
SCHEMBL6916 0.73 BRD4 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2483251-A2 POLYCYCLIC COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS Amira Pharmaceuticals, Inc. (US) 2012-08-08 EP disclosed
WO-2011041462-A2 POLYCYCLIC COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AMIRA PHARMACEUTICALS, INC. (US) 2011-04-07 WO disclosed