SCHEMBL4147159

SCHEMBL4147159

CN(c1nccs1)S(=O)(=O)c1ccc(Nc2nccc(-c3cccc4ccccc34)n2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK9 P50750 9/20 0.51
CCNT1 O60563 8/20 0.51
IKBKB O14920 6/20 0.44
CDK1 P06493 2/20 0.42
CCNB1 P14635 2/20 0.42
SYK P43405 2/20 0.41
GSK3B P49841 3/20 0.41
DKK1 O94907 2/20 0.41
AURKA O14965 1/20 0.41
MAP4K4 O95819 1/20 0.41
ABL1 P00519 1/20 0.41
LCK P06239 1/20 0.41
MET P08581 1/20 0.41
PDGFRB P09619 1/20 0.41
FGFR1 P11362 1/20 0.41
FLT1 P17948 1/20 0.41
KDR P35968 1/20 0.41
FLT3 P36888 1/20 0.41
MAPK8 P45983 1/20 0.41
MAPK9 P45984 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4139765 0.83 IKBKB (0.47) CDK9CCNT1IKBKBCDK1CCNB1
SCHEMBL4146248 0.82 IKBKB (0.56) CDK9CCNT1IKBKBCDK1CCNB1
SCHEMBL4144796 0.81 IKBKB (0.47) CDK9CCNT1IKBKBCDK1CCNB1
SCHEMBL4138290 0.80 CDK2 (0.46) CDK9CCNT1IKBKBCDK1CCNB1
SCHEMBL4151969 0.79 IKBKB (0.51) CDK9CCNT1IKBKBCDK1CCNB1
SCHEMBL3518263 0.76 CDK9 (0.52) CDK9CCNT1IKBKBCDK1CCNB1
SCHEMBL17819109 0.68 DYRK1A (0.49) CDK9CCNT1CDK1CCNB1AURKA
SCHEMBL12522874 0.67 MAPT (0.53)
SCHEMBL4156267 0.67 SYK (0.65) CDK9CCNT1SYKCDK2
SCHEMBL13924521 0.66 SYK (0.65) SYKGSK3BMAPK8CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090048282-A1 PYRIMIDINE SULFONAMIDE ANALOGS AND THEIR USE AS AGONISTS OF THE WNT-BETA-CATENIN CELLULAR MESSAGING SYSTEM WYETH (US) 2009-02-19 US claimed
US-20090048282-A1 PYRIMIDINE SULFONAMIDE ANALOGS AND THEIR USE AS AGONISTS OF THE WNT-BETA-CATENIN CELLULAR MESSAGING SYSTEM WYETH (US) 2009-02-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090048282-A1 PYRIMIDINE SULFONAMIDE ANALOGS AND THEIR USE AS AGONISTS OF THE WNT-BETA-CATENIN CELLULAR MESSAGING SYSTEM WNT1, CTNNB1, WNT3A CDK9 668/4885CCNT1 1400/4885IKBKB 1593/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.