SCHEMBL4146248

SCHEMBL4146248

CN(c1nccs1)S(=O)(=O)c1ccc(Nc2nccc(-c3cc4ccccc4s3)n2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 15/20 0.56
CHUK O15111 9/20 0.56
IKBKG Q9Y6K9 9/20 0.56
MEN1 O00255 1/20 0.46
RECQL P46063 1/20 0.46
BLM P54132 1/20 0.46
KMT2A Q03164 1/20 0.46
PRKCZ Q05513 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
DKK1 O94907 2/20 0.46
GSK3B P49841 2/20 0.46
CCNT1 O60563 3/20 0.44
CDK9 P50750 3/20 0.44
CDK1 P06493 1/20 0.44
CCNB1 P14635 1/20 0.44
CCNA2 P20248 1/20 0.44
CDK2 P24941 1/20 0.44
CDK7 P50613 1/20 0.44
CCNH P51946 1/20 0.44
CCNA1 P78396 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4139765 0.85 IKBKB (0.47) IKBKBMEN1KMT2ADKK1GSK3B
SCHEMBL4151969 0.83 IKBKB (0.51) IKBKBDKK1GSK3BCCNT1CDK9
SCHEMBL4147159 0.82 CDK9 (0.51) IKBKBDKK1GSK3BCCNT1CDK9
SCHEMBL4144796 0.79 IKBKB (0.47) IKBKBDKK1GSK3BCCNT1CDK9
SCHEMBL4138290 0.78 CDK2 (0.46) IKBKBDKK1GSK3BCCNT1CDK9
SCHEMBL3516178 0.78 IKBKB (0.69) IKBKBCHUKIKBKGMEN1RECQL
SCHEMBL4151110 0.74 IKBKB (0.64) IKBKBCHUKIKBKGGSK3BCCNT1
SCHEMBL8308064 0.72 IKBKB (0.82) IKBKBCHUKIKBKGMEN1RECQL
SCHEMBL4148307 0.69 IKBKB (0.58) IKBKBCHUKIKBKGMEN1RECQL
SCHEMBL4146468 0.68 DKK1 (0.52) IKBKBCHUKIKBKGMEN1RECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090048282-A1 PYRIMIDINE SULFONAMIDE ANALOGS AND THEIR USE AS AGONISTS OF THE WNT-BETA-CATENIN CELLULAR MESSAGING SYSTEM WYETH (US) 2009-02-19 US claimed
US-20090048282-A1 PYRIMIDINE SULFONAMIDE ANALOGS AND THEIR USE AS AGONISTS OF THE WNT-BETA-CATENIN CELLULAR MESSAGING SYSTEM WYETH (US) 2009-02-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090048282-A1 PYRIMIDINE SULFONAMIDE ANALOGS AND THEIR USE AS AGONISTS OF THE WNT-BETA-CATENIN CELLULAR MESSAGING SYSTEM WNT1, CTNNB1, WNT3A IKBKB 1593/4885CHUK 584/4885IKBKG 4552/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.