SCHEMBL4149173

SCHEMBL4149173

CN1CCNCC1Cc1ccc(C(=O)O)cc1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.47
CA2 P00918 4/20 0.47
CA4 P22748 4/20 0.47
CA9 Q16790 4/20 0.47
SLC6A2 P23975 4/20 0.46
SLC6A4 P31645 4/20 0.46
SLC6A3 Q01959 4/20 0.46
TDP1 Q9NUW8 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
MITF O75030 1/20 0.41
GRIK1 P39086 2/20 0.41
ALDH1A1 P00352 1/20 0.40
HRH3 Q9Y5N1 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4933217 0.85 MAPT (0.46) CA1CA2CA4CA9ALDH1A1
SCHEMBL4934485 0.82 SLC6A2 (0.47) CA1CA2CA4CA9SLC6A2
SCHEMBL6926417 0.82 SLC6A2 (0.65) CA1CA2CA4CA9SLC6A2
SCHEMBL10413244 0.82 SLC6A2 (0.65) CA1CA2CA4CA9SLC6A2
SCHEMBL22285003 0.82 SLC6A2 (0.65) CA1CA2CA4CA9SLC6A2
SCHEMBL28475644 0.80 SLC6A2 (0.47) SLC6A2SLC6A4SLC6A3TDP1L3MBTL1
SCHEMBL8238773 0.78 PARP1 (0.54) CA1CA2CA4CA9SLC6A2
SCHEMBL12520753 0.77 SLC6A2 (0.44) SLC6A2SLC6A4SLC6A3HRH3
SCHEMBL15557524 0.76 DAO (0.46) CA1CA2CA4CA9SLC6A2
SCHEMBL18600519 0.76 SLC6A4 (0.54) CA1CA2CA4CA9SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117126153-A New coronavirus inhibitor, preparation method, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2023-11-28 CN disclosed
US-20090105259-A1 Acyclic 1,4-Diamines and Uses Thereof SMITHKLINE BEECHAM CORPORATION 2009-04-23 US disclosed
EP-1940785-A2 ACYCLIC 1,4-DIAMINES AND USES THEREOF SmithKline Beecham Corporation (US) 2008-07-09 EP disclosed
WO-2007030761-A2 ACYCLIC 1,4-DIAMINES AND USES THEREOF SMITHKLINE BEECHAM CORPORATION (US) 2007-03-15 WO disclosed
US-7189729-B2 Methods and compositions as protein kinase inhibitors IRM LLC (BM) 2007-03-13 US disclosed
US-20070010529-A1 Nitrogenous heterocyclic compounds and medical use thereof ONO PHARMACEUTICAL CO., LTD. (JP) 2007-01-11 US disclosed
EP-1670771-A1 COMPOUNDS AND COMPOSITIONS AS PROTEIN KINASE INHIBITORS IRM, LLC (BM) 2006-06-21 EP disclosed
US-20050171105-A1 For therapy of benign and malignant proliferative disorders as well as diseases resulting from inappropriate activation of the immune and nervous systems IRM LLC (BM) 2005-08-04 US disclosed
WO-2005033086-A1 COMPOUNDS AND COMPOSITIONS AS PROTEIN KINASE INHIBITORS IRM LLC (BM) 2005-04-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050171105-A1 For therapy of benign and malignant proliferative disorders as well as diseases resulting from inappropriate activation of the immune and nervous systems ERBB2, ERBB3, ERBB4 CA1 4607/4885CA2 2608/4885CA4 3078/4885
US-20070010529-A1 Nitrogenous heterocyclic compounds and medical use thereof MAPK1, NOS1, NOS2 CA1 1486/4885CA2 1212/4885CA4 2114/4885
US-20090105259-A1 Acyclic 1,4-Diamines and Uses Thereof TRPV4, TRPC4, TRPV1 CA1 1033/4885CA2 182/4885CA4 228/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.