Glyoxylate

Glyoxylate

SCHEMBL4152113

O=CC(=O)O.c1ccsc1

nearest known ligand 0.53

Full drug profile on Sugi Atlas →

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.35
MAPK1 P28482 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
HCAR2 Q8TDS4 1/20 0.32
TSHR P16473 2/20 0.30
TP53 P04637 1/20 0.30
EGLN1 Q9GZT9 1/20 0.30
EGLN3 Q9H6Z9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Glyoxylate SCHEMBL1443846 0.97 ALDH1A1 (0.33) ALDH1A1MAPK1TDP1HCAR2
Glyoxylate SCHEMBL27691861 0.97 ALDH1A1 (0.33) ALDH1A1MAPK1TDP1HCAR2
Glyoxylate SCHEMBL28504188 0.97 ALDH1A1 (0.33) ALDH1A1MAPK1TDP1HCAR2
Maleic Acid SCHEMBL27485086 0.82 TSHR (0.53) ALDH1A1HCAR2TSHRTP53EGLN1
Fumaric Acid SCHEMBL10620517 0.82 TSHR (0.53) ALDH1A1HCAR2TSHRTP53EGLN1
Maleic Acid SCHEMBL10620502 0.82 TSHR (0.53) ALDH1A1HCAR2TSHRTP53EGLN1
Thiophene SCHEMBL1616682 0.81
Thiophene SCHEMBL20482064 0.81 CA1 (0.39)
Benzene SCHEMBL4653866 0.80 ALDH1A1 (0.45) ALDH1A1MAPK1TDP1HCAR2TSHR
Thiophene SCHEMBL7050121 0.80 ALDH1A1 (0.32) ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 33 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102245688-B Conductive composite material and thermoelectric device comprising same 3M INNOVATIVE PROPERTIES CO 2014-03-12 CN claimed
CN-101880271-B Synthesis method of 2-thiophene acetylchloride Lianyungang hongye chemical industry co ltd 2012-11-28 CN claimed
CN-102245688-A Conductive composite material and thermoelectric device comprising same 3M INNOVATIVE PROPERTIES CO 2011-11-16 CN claimed
CN-101880271-A Synthesis method of 2-thiophene acetylchloride Lianyungang hongye chemical industry co ltd 2010-11-10 CN claimed
US-20090209465-A1 MCT1 Transporters Expressed in Blood Brain Barrier Cells XENOPORT, INC. (US) 2009-08-20 US claimed
US-7452680-B2 Using monocarboxylate transporter 1 (MCT1) as diagnostic tool in detecting modulators for prevention and treatment of nervous system disorders XENOPORT, INC. (US) 2008-11-18 US claimed
WO-2005075992-A1 MCT1 TRANSPORTER EXPRESSED IN BLOOD BRAIN BARRIER CELLS XENOPORT, INC. (US) 2005-08-18 WO claimed
US-20050170390-A1 MCT1 transporters expressed in blood brain barrier cells XENOPORT, INC. (US) 2005-08-04 US claimed
US-20240208895-A1 BRANCHED-CHAIN AMINO ACID DERIVATIVES TO TREAT DISEASE Intrabio Ltd. (GB) 2024-06-27 US disclosed
CN-118184625-A Synthesis method of 2-thiopheneacetic acid 浙江东盈药业有限公司 2024-06-14 CN disclosed
WO-2022264037-A1 BRANCHED-CHAIN AMINO ACID DERIVATIVES TO TREAT DISEASE Intrabio Ltd. (GB) 2022-12-22 WO disclosed
CN-113552782-A Light-responsive material, adhesive, photoswitch material, toner, and image forming method 柯尼卡美能达株式会社 2021-10-26 CN disclosed
CN-103992302-A Synthesis process of 2-thiopheneacetic acid SHANGQIU KOREATA CHEMICAL CO LTD 2014-08-20 CN disclosed
CN-102977073-B Method for synthesizing 2-thiophene acetic acid through 2-thiophene alcohol UNIV SHANDONG NORMAL 2014-05-14 CN disclosed
WO-2005098444-A2 MONOCARBOXYLATE TRANSPORTERS EXPRESSED IN CANCER CELLS XENOPORT, INC. (US) 2005-10-20 WO disclosed
WO-2005075992-A1 MCT1 TRANSPORTER EXPRESSED IN BLOOD BRAIN BARRIER CELLS XENOPORT, INC. (US) 2005-08-18 WO disclosed
US-20050170390-A1 MCT1 transporters expressed in blood brain barrier cells XENOPORT, INC. (US) 2005-08-04 US disclosed
US-20050032135-A1 Monocarboxylate transporters expressed in cancer cells XENOPORT, INC. (US) 2005-02-10 US disclosed
CN-1382140-A Neurotrophic pyrrolidines and piperidines and related compositions containing them ORTHO MCNEIL PHARM INC (US) 2002-11-27 CN disclosed
US-4369206-A HARDENING COATING WITH AMINES BAYER AKTIENGESELLSCHAFT (DE) 1983-01-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050032135-A1 Monocarboxylate transporters expressed in cancer cells SLC16A1, SLC16A3, SLC16A8 ALDH1A1 523/4885MAPK1 3089/4885TDP1 3152/4885
US-20240208895-A1 BRANCHED-CHAIN AMINO ACID DERIVATIVES TO TREAT DISEASE CTSA, GBA1, GAA ALDH1A1 2303/4885MAPK1 3010/4885TDP1 635/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.