SCHEMBL4157933

SCHEMBL4157933

CN(C(=O)c1c(F)cccc1F)C(=O)N(C)c1ccc(S(=O)(=O)C(F)(F)C(F)F)cc1F

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 2/20 0.35
TDP1 Q9NUW8 1/20 0.34
RORC P51449 3/20 0.34
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
GPBAR1 Q8TDU6 3/20 0.31
TLR7 Q9NYK1 1/20 0.31
POLB P06746 1/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4144866 0.89 EPAS1 (0.39) SIRT2TDP1RORCALDH1A1CYP3A4
SCHEMBL4150636 0.82 KMT2A (0.36) SIRT2TDP1RORCCYP3A4CYP2C9
SCHEMBL4915675 0.81 TLR7 (0.38) TDP1RORCTLR7POLBMEN1
SCHEMBL4150845 0.78 RORC (0.35) TDP1RORCTLR7POLB
SCHEMBL4151440 0.77 RORC (0.34) TDP1RORCGPBAR1TLR7POLB
SCHEMBL4913480 0.77 TLR7 (0.44) TDP1RORCALDH1A1GPBAR1TLR7
SCHEMBL4636520 0.76 KAT6A (0.38) SIRT2GPBAR1POLB
SCHEMBL4153993 0.75 RORC (0.37) SIRT2TDP1RORCGPBAR1TLR7
SCHEMBL13774593 0.74 RORC (0.39) SIRT2TDP1RORCTLR7POLB
SCHEMBL4154435 0.74 RORC (0.36) SIRT2TDP1RORCGPBAR1TLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090176786-A1 Benzoylurea Compounds and Use Thereof SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2009-07-09 US disclosed
US-20090176786-A1 Benzoylurea Compounds and Use Thereof SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2009-07-09 US disclosed
EP-1937629-A2 BENZOYLUREA COMPOUNDS AND USE THEREOF Sumitomo Chemical Company, Limited (JP) 2008-07-02 EP disclosed
WO-2007046513-A2 BENZOYLUREA COMPOUNDS AND USE THEREOF SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2007-04-26 WO disclosed
WO-2007046513-A2 BENZOYLUREA COMPOUNDS AND USE THEREOF SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2007-04-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090176786-A1 Benzoylurea Compounds and Use Thereof BTK, BRIX1, NFXL1 SIRT2 2533/4885TDP1 1690/4885RORC 4448/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.