SCHEMBL4158191

SCHEMBL4158191

NS(=O)(=O)c1c(NC(=O)c2cnc3c(C(F)(F)F)cccc3c2)cccc1-c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.44
SCN5A Q14524 6/20 0.44
SCN9A Q15858 6/20 0.44
LCK P06239 4/20 0.42
KDR P35968 4/20 0.42
MAPK14 Q16539 4/20 0.42
JAK3 P52333 3/20 0.42
BRAF P15056 1/20 0.41
NTRK1 P04629 6/20 0.41
RXFP1 Q9HBX9 1/20 0.41
NTRK3 Q16288 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4165746 0.90 ALDH1A1 (0.44) ALDH1A1SCN5ASCN9ALCKKDR
SCHEMBL4158189 0.72 PARP1 (0.43) SCN9A
SCHEMBL4306073 0.71 NR1H2 (0.37)
SCHEMBL28235432 0.71 PSMD14 (0.60)
SCHEMBL11499102 0.70 HPGDS (0.54) BRAF
SCHEMBL7451848 0.70 PSMD14 (0.61) SCN9A
SCHEMBL2452806 0.70 CA1 (0.41) SCN9A
SCHEMBL10871494 0.69 PSMD14 (0.69)
SCHEMBL31124478 0.67 PSMD14 (0.43) BRAF
SCHEMBL17934555 0.67 ALDH1A1 (0.61) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed