SCHEMBL4158549

SCHEMBL4158549

COc1cc(-c2cnc(N)c(-c3nc4ccccc4n3CCN3CCOCC3)n2)ccc1OCCN1CCOCC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP3K11 Q16584 2/20 0.50
KDM4E B2RXH2 3/20 0.47
HSD17B10 Q99714 2/20 0.47
RECQL P46063 1/20 0.47
JAK2 O60674 6/20 0.47
JAK1 P23458 6/20 0.47
JAK3 P52333 5/20 0.47
KIT P10721 1/20 0.45
EGFR P00533 2/20 0.45
LMNA P02545 1/20 0.44
ALDH1A1 P00352 2/20 0.44
TP53 P04637 2/20 0.44
MAPT P10636 1/20 0.44
GAA P10253 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
TYK2 P29597 4/20 0.43
PDPK1 O15530 1/20 0.43
ADORA2A P29274 1/20 0.43
NPC1 O15118 1/20 0.42
HPGD P15428 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4010236 0.94 JAK2 (0.51) MAP3K11KDM4EHSD17B10RECQLJAK2
SCHEMBL3924773 0.86 EGFR (0.48) KDM4EHSD17B10RECQLJAK2JAK1
SCHEMBL3928126 0.85 MCHR1 (0.47) MAP3K11KDM4EHSD17B10RECQLADORA2A
SCHEMBL4297778 0.82 ATR (0.58) MAP3K11JAK2JAK1JAK3KIT
SCHEMBL4139890 0.82 KDM4E (0.50) KDM4EHSD17B10RECQLEGFRALDH1A1
SCHEMBL4006573 0.75 ATR (0.59) EGFR
SCHEMBL2801860 0.75 JAK2 (0.59) MAP3K11JAK2JAK1JAK3KIT
SCHEMBL18832177 0.72 KIT (0.59) MAP3K11KITPDPK1ADORA2A
SCHEMBL30505753 0.72 KIT (0.59) MAP3K11KITPDPK1ADORA2A
SCHEMBL2799644 0.71 JAK2 (0.64) MAP3K11KDM4EJAK2JAK1JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007390-A2 2-PYRAZ INYLBENZ IMIDAZOLE DERIVATIVES AS RECEPTOR TYROSINE KINASE INHIBITORS ASTRAZENECA AB (SE) 2009-01-15 WO claimed