SCHEMBL4159925

SCHEMBL4159925

O=C(Cc1ccsc1)N[C@@H](CCCSCC(=O)C(F)(F)F)C(=O)NCCc1c[nH]c2ccccc12

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.45
MEN1 O00255 3/20 0.45
ALDH1A1 P00352 2/20 0.45
MAPT P10636 2/20 0.45
KDM4E B2RXH2 1/20 0.45
CYP3A4 P08684 1/20 0.45
ALOX15 P16050 1/20 0.45
TSHR P16473 1/20 0.45
MAPK1 P28482 1/20 0.45
HSD17B10 Q99714 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
BRS3 P32247 2/20 0.43
CTSC P53634 1/20 0.43
NMBR P28336 5/20 0.42
USP2 O75604 1/20 0.42
TACR3 P29371 1/20 0.41
HSD17B2 P37059 1/20 0.41
TACR1 P25103 1/20 0.41
GOT1 P17174 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4605724 0.86 CES1 (0.46)
SCHEMBL5125744 0.80 MTNR1A (0.50) KMT2AMEN1ALDH1A1MAPTKDM4E
SCHEMBL4153988 0.78 L3MBTL1 (0.47) KMT2AMEN1ALDH1A1CTSCNMBR
SCHEMBL4174445 0.78 HDAC1 (0.42) KMT2AMEN1ALDH1A1MAPTKDM4E
SCHEMBL4159928 0.77 MC5R (0.39)
SCHEMBL4174440 0.76 SHMT1 (0.41) ALDH1A1KDM4E
Trifluoroacetic Acid SCHEMBL4163740 0.74 MCHR1 (0.41)
SCHEMBL4174424 0.74 SIGMAR1 (0.38) KMT2AMEN1ALDH1A1MAPT
SCHEMBL4166185 0.73 NPC1 (0.42) KMT2AMEN1ALDH1A1MAPTCYP3A4
Trifluoroacetic Acid SCHEMBL4169498 0.71 HDAC4 (0.39) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090054448-A1 Amino Acid Derivatives as Histone Deacetylase (HDAC) Inhibitors JONES PHILIP 2009-02-26 US disclosed
EP-1945609-A2 AMINO ACID DERIVATIVES AS HISTONE DEACETYLASE (HDAC) INHIBITORS ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI S.P.A. (IT) 2008-07-23 EP disclosed
WO-2007029036-A2 AMINO ACID DERIVATIVES AS HISTONE DEACETYLASE (HDAC) INHIBITORS ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2007-03-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090054448-A1 Amino Acid Derivatives as Histone Deacetylase (HDAC) Inhibitors HDAC5, HDAC1, HDAC11 KMT2A 20/4885MEN1 3953/4885ALDH1A1 320/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.