Trifluoroacetic Acid

Trifluoroacetic Acid

SCHEMBL4161040

NC(=O)[C@H](CCCSCC(=O)C(F)(F)F)N(C(=O)Cc1ccsc1)C1CCN(Cc2ccccc2)CC1.O=C(O)C(F)(F)F

nearest known ligand 0.43

Full drug profile on Sugi Atlas →

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 5/20 0.43
OPRM1 P35372 6/20 0.42
OPRD1 P41143 4/20 0.42
OPRK1 P41145 4/20 0.42
KCNH2 Q12809 1/20 0.40
CHRM2 P08172 4/20 0.38
CHRM3 P20309 4/20 0.38
CES1 P23141 1/20 0.35
SLC2A1 P11166 1/20 0.35
CHRM1 P11229 1/20 0.34
CPB2 Q96IY4 1/20 0.34
DRD2 P14416 1/20 0.33
DRD4 P21917 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL4606076 0.93 KCNH2 (0.46) SIGMAR1OPRM1KCNH2CHRM2CHRM3
SCHEMBL4174427 0.86 SIGMAR1 (0.36) SIGMAR1OPRM1OPRD1OPRK1CES1
Trifluoroacetic Acid SCHEMBL4164046 0.86 SLC2A1 (0.40) SIGMAR1OPRM1OPRD1OPRK1KCNH2
Trifluoroacetic Acid SCHEMBL4166752 0.85 KCNH2 (0.39) SIGMAR1OPRM1OPRD1KCNH2CHRM2
Trifluoroacetic Acid SCHEMBL4159827 0.84 BCHE (0.42) KCNH2CHRM2CHRM3CES1SLC2A1
Trifluoroacetic Acid SCHEMBL4156617 0.84 ACHE (0.41) KCNH2SLC2A1DRD2DRD4
Trifluoroacetic Acid SCHEMBL4154008 0.82 CHRM2 (0.38) SIGMAR1OPRM1KCNH2CHRM2CHRM3
Trifluoroacetic Acid SCHEMBL4622705 0.80 ALDH1A1 (0.39) CHRM1
Trifluoroacetic Acid SCHEMBL4171441 0.80 CHRM3 (0.42) SIGMAR1CHRM2CHRM3
Trifluoroacetic Acid SCHEMBL4161039 0.77 SIGMAR1 (0.57) SIGMAR1CHRM2CHRM3CHRM1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090054448-A1 Amino Acid Derivatives as Histone Deacetylase (HDAC) Inhibitors JONES PHILIP 2009-02-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090054448-A1 Amino Acid Derivatives as Histone Deacetylase (HDAC) Inhibitors HDAC5, HDAC1, HDAC11 SIGMAR1 3623/4885OPRM1 3936/4885OPRD1 3774/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.