SCHEMBL416168

SCHEMBL416168

COC(=O)c1ccc(C(F)(F)C(F)(F)F)c(F)c1C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CFTR P13569 3/20 0.41
NPC1 O15118 1/20 0.38
CASP3 P42574 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
SENP8 Q96LD8 1/20 0.38
SENP7 Q9BQF6 1/20 0.38
SENP6 Q9GZR1 1/20 0.38
NOTUM Q6P988 1/20 0.38
SOS1 Q07889 1/20 0.38
MYC P01106 2/20 0.37
PDK2 Q15119 2/20 0.37
PDK4 Q16654 2/20 0.37
CA12 O43570 2/20 0.37
CA1 P00915 2/20 0.37
CA2 P00918 2/20 0.37
CA7 P43166 2/20 0.37
CA9 Q16790 2/20 0.37
CA14 Q9ULX7 2/20 0.37
SLC6A4 P31645 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL417766 0.83 TAS2R14 (0.38) NOTUMMYCTSHRKDM4EALDH1A1
SCHEMBL416274 0.81 CFTR (0.38) CFTRNPC1CASP3RAB9ASMN1; SMN2
SCHEMBL1235475 0.78 CFTR (0.46) CFTRNPC1CASP3RAB9ASMN1; SMN2
SCHEMBL30720952 0.76 CES2 (0.50) CFTRNPC1CASP3RAB9ASMN1; SMN2
SCHEMBL8217125 0.76 CES2 (0.50) CFTRNPC1CASP3RAB9ASMN1; SMN2
SCHEMBL25269151 0.75 CFTR (0.44) CFTRNOTUMPDK2PDK4CA12
SCHEMBL30230910 0.75 CFTR (0.44) CFTRNOTUMPDK2PDK4CA12
SCHEMBL30966098 0.75 CA1 (0.50) CFTRNPC1CASP3RAB9ASMN1; SMN2
SCHEMBL25475896 0.75 CA1 (0.50) CFTRNPC1CASP3RAB9ASMN1; SMN2
SCHEMBL22831692 0.73 CFTR (0.49) CFTRNPC1CASP3RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8603947-B2 (4-haloalkyl-3-thiobenzoyl)cyclohexanediones and use thereof as herbicides BAYER CROPSCIENCE AG (DE) 2013-12-10 US disclosed
US-8536097-B2 4-(4-haloalkyl-3-thiobenzoyl)pyrazoles and use thereof as herbicides BAYER CROPSCIENCE AG (DE) 2013-09-17 US disclosed
US-20120021904-A1 (4-HALOALKYL-3-THIOBENZOYL)CYCLOHEXANEDIONES AND USE THEREOF AS HERBICIDES BAYER CROPSCIENCE AG (DE) 2012-01-26 US disclosed
US-20120021903-A1 4-(4-HALOALKYL-3-THIOBENZOYL)PYRAZOLES AND USE THEREOF AS HERBICIDES BAYER CROPSCIENCE AG (DE) 2012-01-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120021904-A1 (4-HALOALKYL-3-THIOBENZOYL)CYCLOHEXANEDIONES AND USE THEREOF AS HERBICIDES CBR3, CBR1, CYP8B1 CFTR 988/4885NPC1 4637/4885CASP3 619/4885
US-20120021903-A1 4-(4-HALOALKYL-3-THIOBENZOYL)PYRAZOLES AND USE THEREOF AS HERBICIDES CBR3, CYP4X1, PRDX4 CFTR 958/4885NPC1 4800/4885CASP3 282/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.