SCHEMBL4173014

SCHEMBL4173014

O=S(=O)(Nc1nccs1)c1ccc(CNCc2ccc(OC(F)(F)F)c(F)c2)cc1F

nearest known ligand 0.66

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 14/20 0.66
SCN3A Q9NY46 5/20 0.66
SCN1A P35498 5/20 0.66
SCN5A Q14524 5/20 0.66
SCN8A Q9UQD0 5/20 0.66
SCN2A Q99250 2/20 0.66
SCN10A Q9Y5Y9 2/20 0.66
KCNH2 Q12809 1/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3161008 0.88 SCN3A (0.86) SCN9ASCN3ASCN1ASCN5ASCN8A
SCHEMBL3173728 0.82 SCN3A (0.82) SCN9ASCN3ASCN1ASCN5ASCN8A
SCHEMBL3167092 0.80 SCN3A (0.83) SCN9ASCN3ASCN1ASCN5ASCN8A
SCHEMBL3119441 0.80 SCN3A (1.00) SCN9ASCN3ASCN1ASCN5ASCN8A
SCHEMBL3168686 0.80 SCN3A (0.82) SCN9ASCN3ASCN1ASCN5ASCN8A
SCHEMBL3066948 0.79 SCN3A (0.66) SCN9ASCN3ASCN1ASCN5ASCN8A
SCHEMBL3160028 0.78 SCN3A (0.67) SCN9ASCN3ASCN1ASCN5ASCN8A
SCHEMBL3165510 0.78 SCN3A (0.69) SCN9ASCN3ASCN1ASCN5ASCN8A
SCHEMBL3166158 0.76 SCN3A (0.78) SCN9ASCN3ASCN1ASCN5ASCN8A
SCHEMBL712204 0.75 ALPL (0.59) SCN9ASCN3ASCN1ASCN5ASCN8A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8357711-B2 Heterocyclic sulfonamides as inhibitors of ion channels PFIZER LIMITED (GB) 2013-01-22 US disclosed
US-20090143358-A1 INHIBITORS OF ION CHANNELS ICAGEN, INC. (US) 2009-06-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090143358-A1 INHIBITORS OF ION CHANNELS TRPV1, TRPV5, TRPA1 SCN9A 51/4885SCN3A 13/4885SCN1A 6/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.