⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.
Similar compounds — the chemically nearest patent molecules
Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.
| Compound | similarity | top predicted | shared targets | |
|---|---|---|---|---|
| SCHEMBL28490272 | 0.97 | CES2 (0.44) | — | |
| SCHEMBL9080757 | 0.78 | LTA4H (0.52) | — | |
| SCHEMBL810985 | 0.78 | — | — | |
| SCHEMBL38016 | 0.76 | DPP4 (0.50) | — | |
| SCHEMBL7527333 | 0.75 | — | — | |
| SCHEMBL6253138 | 0.75 | CES2 (0.41) | — | |
| SCHEMBL27991580 | 0.73 | DPP4 (0.47) | — | |
| SCHEMBL832620 | 0.73 | — | — | |
| SCHEMBL28995862 | 0.73 | DPP4 (0.47) | — | |
| SCHEMBL28167953 | 0.73 | DPP4 (0.47) | — |
Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.
Patent provenance — the patents this molecule appears in, and who filed them
Claimed or disclosed in 159 patents. claimed = in the patent's claims; disclosed = body only.
| Patent | Title | Assignee | Published | Priority | Filing | Country | Status |
|---|---|---|---|---|---|---|---|
| CN-106632065-B | Benzimidazoles compound and its application | 沈阳药科大学 | 2019-08-30 | — | — | CN | claimed |
| CN-108164408-A | A kind of novel synthesis of 7- halogen -1- indones | 常熟浸大科技有限公司 | 2018-06-15 | — | — | CN | claimed |
| CN-106632065-A | Benzimidazole compound and application thereof | 沈阳药科大学 | 2017-05-10 | — | — | CN | claimed |
| CN-104961665-B | Cool compound of six benzos of dovetail shaped side chain Sulfide-containing Hindered and preparation method thereof | 北京印刷学院 | 2017-03-01 | — | — | CN | claimed |
| CN-104961665-A | Hexabenzocoronene compound containing thioether in dovetail-like side-chain and preparation method thereof | BEIJING INST GRAPHIC COMM | 2015-10-07 | — | — | CN | claimed |
| JP-4642766-B2 | — | — | 2011-03-02 | — | — | JP | claimed |
| US-7589086-B2 | Substituted pyrazolo[3,4-D]pyrimidines as anti-tumor agents | UNIVERSITA DEGLI STUDI DI SIENA (IT) | 2009-09-15 | — | — | US | claimed |
| EP-1638966-B1 | 4-SUBSTITUTED DERIVATIVES OF PYRAZOLO ¬3,4-d PYRIMIDINE AND USES THEREOF | UNIV SIENA (IT) | 2008-03-19 | — | — | EP | claimed |
| JP-2007501861-A | — | — | 2007-02-01 | — | — | JP | claimed |
| JP-2007500206-A | — | — | 2007-01-11 | — | — | JP | claimed |
| US-20070010510-A1 | 4-Substituted derivatives of pyrazolo[3,4-d]pyrimidine and pyrrolo[2,3-d]pyrimidine and uses thereof | UNIVERSITA DEGLI STUDI DI SIENA (IT) | 2007-01-11 | — | — | US | claimed |
| EP-1651229-A1 | GUANIDINO-SUBSTITUTED QUINAZOLINONE COMPOUNDS AS MC4-R AGONISTS | Chiron Corporation (US) | 2006-05-03 | — | — | EP | claimed |
| EP-1638966-A2 | 4-SUBSTITUTED DERIVATIVES OF PYRAZOLO ¬3,4-d| PYRIMIDINE AND PYRROLO ¬2,3-d| PYRIMIDINE AND USES THEREOF | UNIVERSITA DEGLI STUDI DI SIENA (IT) | 2006-03-29 | — | — | EP | claimed |
| WO-2004112793-A1 | GUANIDINO-SUBSTITUTED QUINAZOLINONE COMPOUNDS AS MC4-R AGONISTS | CHIRON CORPORATION (US) | 2004-12-29 | — | — | WO | claimed |
| WO-2004106340-A2 | 4-SUBSTITUTED DERIVATIVES OF PYRAZOLO [3,4-d] PYRIMIDINE AND PYRROLO [2,3-d] PYRIMIDINE AND USES THEREOF | UNIVERSITÀ DEGLI STUDI DI SIENA (IT) | 2004-12-09 | — | — | WO | claimed |
| US-6235928-B1 | ENZYME INHIBITOR MATRIX METALLOPROTEINASE FAMILY, INCLUDING COLLAGENASE, STROMELYSIN, AND GELATINASE, THE COMPOUNDS OR PHARMACEUTICAL COMPOSITIONS | PHARMACIA & UPJOHN COMPANY | 2001-05-22 | — | — | US | claimed |
| EP-0929519-A1 | $g(b)-SULFONYL HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASES INHIBITORS | PHARMACIA & UPJOHN COMPANY (US) | 1999-07-21 | — | — | EP | claimed |
| US-5847153-A | β-sulfonyl hydroxamic acids | PHARMACIA & UPJOHN COMPANY (US) | 1998-12-08 | — | — | US | claimed |
| WO-1998013340-A1 | β-SULFONYL HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASES INHIBITORS | PHARMACIA & UPJOHN COMPANY (US) | 1998-04-02 | — | — | WO | claimed |
| CN-117777773-A | Active energy ray-curable composition, cured product, and film | DIC株式会社 | 2024-03-29 | — | — | CN | disclosed |
| CN-117777774-A | Active energy ray-curable composition, cured product, and film | DIC株式会社 | 2024-03-29 | — | — | CN | disclosed |
| CN-110959202-B | Composition for encapsulating organic light emitting diode and organic light emitting diode display | 三星SDI株式会社 | 2023-08-25 | — | — | CN | disclosed |
| CN-109952663-B | Composition for sealing organic light-emitting element and organic light-emitting element display device manufactured from the same | 三星SDI株式会社 | 2023-07-21 | — | — | CN | disclosed |
| CN-110769821-B | Spiro indolines as IL-17 modulators | UCB生物制药有限责任公司 | 2023-07-07 | — | — | CN | disclosed |
| US-20230203225-A1 | COMPOSITION FOR ENCAPSULATING ORGANIC LIGHT EMITTING ELEMENT AND ORGANIC LIGHT EMITTING ELEMENT DISPLAY DEVICE MANUFACTURED THEREFROM | SAMSUNG SDI CO LTD (KR) | 2023-06-29 | — | — | US | disclosed |
| CN-111465662-B | Aqueous dispersion of coloured particles | 三菱铅笔株式会社 | 2023-05-26 | — | — | CN | disclosed |
| US-20230151246-A1 | ADHESIVE COMPOSITION, ADHESIVE LAYER FORMED THEREFROM, AND OPTICAL DISPLAY DEVICE COMPRISING SAME | SAMSUNG SDI CO., LTD. (KR) | 2023-05-18 | — | — | US | disclosed |
| CN-115916918-A | Adhesive composition, adhesive layer formed therefrom, and optical display device comprising same | 三星SDI株式会社 | 2023-04-04 | — | — | CN | disclosed |
| US-20230102431-A1 | COMPOSITION FOR ORGANIC LIGHT EMITTING DIODE ENCAPSULATION AND ORGANIC LIGHT EMITTING DIODE DISPLAY MANUFACTURED THEREFROM | SAMSUNG SDI CO., LTD. (KR) | 2023-03-30 | — | — | US | disclosed |
| US-11608400-B2 | Composition for encapsulating organic light emitting element and organic light emitting element display device manufactured therefrom | SAMSUNG SDI CO., LTD. (KR) | 2023-03-21 | — | — | US | disclosed |
| CN-115722238-A | Method for synthesizing olefin monomer by catalytic conversion of biomass glycosyl compound and preparation of reversible solidified liquid rubber | 中国科学院长春应用化学研究所 | 2023-03-03 | — | — | CN | disclosed |
| US-20230006135-A1 | COMPOSITION FOR ENCAPSULATING ORGANIC LIGHT EMITTING DIODE AND ORGANIC LIGHT EMITTING DIODE DISPLAY COMPRISING ORGANIC LAYER FORMED USING THE SAME | SAMSUNG SDI CO., LTD. (KR) | 2023-01-05 | — | — | US | disclosed |
| US-11539025-B2 | Composition for organic light emitting diode encapsulation and organic light emitting diode display manufactured therefrom | SAMSUNG SDI CO., LTD. (KR) | 2022-12-27 | — | — | US | disclosed |
| CN-110872365-B | Composition for encapsulating organic light emitting diode and organic light emitting diode display | 三星SDI株式会社 | 2022-04-15 | — | — | CN | disclosed |
| CN-113454132-A | Ultraviolet-absorbing polymer, resin composition for molding, and molded article | 东洋油墨SC控股株式会社 | 2021-09-28 | — | — | CN | disclosed |
| CN-113248653-A | Composition for encapsulating organic light emitting device and organic light emitting device display apparatus | 三星SDI株式会社 | 2021-08-13 | — | — | CN | disclosed |
| US-11052076-B2 | Spirocyclic indolines as IL-17 modulators | UCB Biopharma SRL (BE) | 2021-07-06 | — | — | US | disclosed |
| US-20210151713-A1 | COMPOSITION FOR ORGANIC LIGHT EMITTING DIODE ENCAPSULATION AND ORGANIC LIGHT EMITTING DIODE DISPLAY MANUFACTURED THEREFROM | SAMSUNG SDI CO., LTD. (KR) | 2021-05-20 | — | — | US | disclosed |
| CN-106715487-B | Process for producing olefin (co) polymer containing constituent unit derived from 1-butene | 三井化学株式会社 | 2021-02-26 | — | — | CN | disclosed |
| CN-108473784-B | Polyfunctional polymerizable compound and coloring composition | 富士胶片和光纯药株式会社 | 2021-01-12 | — | — | CN | disclosed |
| CN-108137755-B | Composition for encapsulating organic light emitting element and organic light emitting element display device manufactured therefrom | 三星SDI株式会社 | 2020-10-20 | — | — | CN | disclosed |
| CN-111465662-A | Aqueous dispersions of pigmented particles | 三菱铅笔株式会社 | 2020-07-28 | — | — | CN | disclosed |
| US-20200138797-A1 | Spirocyclic Indolines as IL-17 Modulators | UCB Biopharma SRL (BE) | 2020-05-07 | — | — | US | disclosed |
| EP-3638227-A1 | SPIROCYCLIC INDOLINES AS IL-17 MODULATORS | UCB Biopharma SRL (BE) | 2020-04-22 | — | — | EP | disclosed |
| CN-110959202-A | Composition for encapsulating organic light emitting diode element and organic light emitting diode display prepared using the same | 三星SDI株式会社 | 2020-04-03 | — | — | CN | disclosed |
| CN-110872365-A | Composition for encapsulating organic light emitting diode and organic light emitting diode display | 三星SDI株式会社 | 2020-03-10 | — | — | CN | disclosed |
| CN-110769821-A | Spirocyclic indolines as IL-17 modulators | UCB生物制药私人有限公司 | 2020-02-07 | — | — | CN | disclosed |
| CN-106632065-B | Benzimidazoles compound and its application | 沈阳药科大学 | 2019-08-30 | — | — | CN | disclosed |
| CN-107452889-B | Composition for encapsulating organic light emitting device and the organic light emitting display using it | 三星SDI株式会社 | 2019-08-13 | — | — | CN | disclosed |
| CN-106257682-B | Organic light emitting diode display equipment | 三星SDI株式会社 | 2019-07-23 | — | — | CN | disclosed |
| CN-110003042-A | α, α -difluoroallyl aromatic hydrocarbon compound and preparation method thereof | 南京工业大学 | 2019-07-12 | — | — | CN | disclosed |
| CN-109952663-A | Organic illuminating element composition for sealing and the organic illuminating element display device as manufactured by the composition | 三星SDI株式会社 | 2019-06-28 | — | — | CN | disclosed |
| CN-106232685-B | Constituent for encapsulating organic light emitting diode and the display using its preparation | 三星SDI株式会社 | 2019-06-21 | — | — | CN | disclosed |
| US-10319946-B2 | Organic light emitting device encapsulating composition, and organic light emitting device display apparatus manufactured using same | SAMSUNG SDI CO., LTD. (KR) | 2019-06-11 | — | — | US | disclosed |
| CN-106257681-B | Organic light emitting diode display equipment | 三星SDI株式会社 | 2019-06-11 | — | — | CN | disclosed |
| CN-106459558-B | Hardening resin composition, its solidfied material, semiconductor-encapsulating material, semiconductor device, prepreg, circuit substrate, laminated film | DIC株式会社 | 2019-03-08 | — | — | CN | disclosed |
| WO-2018229079-A1 | SPIROCYCLIC INDOLINES AS IL-17 MODULATORS | UCB BIOPHARMA SPRL (BE) | 2018-12-20 | — | — | WO | disclosed |
| US-20180342674-A1 | COMPOSITION FOR ENCAPSULATING ORGANIC LIGHT EMITTING ELEMENT AND ORGANIC LIGHT EMITTING ELEMENT DISPLAY DEVICE MANUFACTURED THEREFROM | SAMSUNG SDI CO., LTD. (KR) | 2018-11-29 | — | — | US | disclosed |
| CN-108473784-A | Polyfunctional polymerizable compound and coloring composition | 富士胶片和光纯药株式会社 | 2018-08-31 | — | — | CN | disclosed |
| CN-108164408-A | A kind of novel synthesis of 7- halogen -1- indones | 常熟浸大科技有限公司 | 2018-06-15 | — | — | CN | disclosed |
| CN-108137755-A | COMPOSITION FOR ENCAPSULATING ORGANIC LIGHT EMITTING ELEMENT AND ORGANIC LIGHT EMITTING ELEMENT DISPLAY DEVICE MANUFACTURED THEREFROM | 三星SDI株式会社 | 2018-06-08 | — | — | CN | disclosed |
| US-9847510-B2 | Organic light emitting diode display apparatus | SAMSUNG SDI CO., LTD. (KR) | 2017-12-19 | — | — | US | disclosed |
| CN-107452889-A | For encapsulating organic light emitting device composition and use its OLED | 三星SDI株式会社 | 2017-12-08 | — | — | CN | disclosed |
| US-9837633-B2 | Organic light emitting diode display apparatus | SAMSUNG SDI CO., LTD. (KR) | 2017-12-05 | — | — | US | disclosed |
| CN-105143279-B | The manufacture method and catalyst for olefines polymerizing of olefin polymer | 三井化学株式会社 | 2017-10-27 | — | — | CN | disclosed |
| US-20170149016-A1 | ORGANIC LIGHT EMITTING DEVICE ENCAPSULATING COMPOSITION, AND ORGANIC LIGHT EMITTING DEVICE DISPLAY APPARATUS MANUFACTURED USING SAME | SAMSUNG SDI CO., LTD. (KR) | 2017-05-25 | — | — | US | disclosed |
| CN-106715487-A | Method for producing olefin (co)polymer containing constituent unit derived from 1-butene | 三井化学株式会社 | 2017-05-24 | — | — | CN | disclosed |
| CN-106632065-A | Benzimidazole compound and application thereof | 沈阳药科大学 | 2017-05-10 | — | — | CN | disclosed |
| CN-104961665-B | Cool compound of six benzos of dovetail shaped side chain Sulfide-containing Hindered and preparation method thereof | 北京印刷学院 | 2017-03-01 | — | — | CN | disclosed |
| CN-106459558-A | Curable resin composition, cured product thereof, semiconductor sealing material, semiconductor device, prepreg, circuit board, and buildup film | DIC株式会社 | 2017-02-22 | — | — | CN | disclosed |
| CN-106257681-A | Organic light emitting diode display equipment | 三星SDI株式会社 | 2016-12-28 | — | — | CN | disclosed |
| CN-106257682-A | Organic light emitting diode display equipment | 三星SDI株式会社 | 2016-12-28 | — | — | CN | disclosed |
| US-20160372704-A1 | ORGANIC LIGHT EMITTING DIODE DISPLAY APPARATUS | SAMSUNG SDI CO., LTD. (KR) | 2016-12-22 | — | — | US | disclosed |
| US-20160372707-A1 | ORGANIC LIGHT EMITTING DIODE DISPLAY APPARATUS | SAMSUNG SDI CO., LTD. (KR) | 2016-12-22 | — | — | US | disclosed |
| CN-106232685-A | Organic luminescent assembly encapsulates constituent and uses its organic luminescent assembly display device prepared | 三星SDI株式会社 | 2016-12-14 | — | — | CN | disclosed |
| CN-104961665-A | Hexabenzocoronene compound containing thioether in dovetail-like side-chain and preparation method thereof | BEIJING INST GRAPHIC COMM | 2015-10-07 | — | — | CN | disclosed |
| CN-101218203-B | Fluorinated derivatives of 4- (2-amino-1-hydroxyethyl) phenol as beta 2 adrenoreceptor agonists | ALMIRALL SA | 2012-05-30 | — | — | CN | disclosed |
| US-20120022048-A1 | Anti-proliferative substituted pyrazolo[3,4-d]pyrimidines derivatives (SPP) to inhibit immune activation, virus replication and tumor growth | LORI FRANCO (US) | 2012-01-26 | — | — | US | disclosed |
| CN-102282234-A | Material for organic electroluminescent device | — | 2011-12-14 | — | — | CN | disclosed |
| WO-2011014239-A1 | ANTI-PROLIFERATIVE SUBSTITUTED PYRAZOLO[3,4-D]PYRIMIDINES DERIVATIVES (SPP) TO INHIBIT IMMUNE ACTIVATION, VIRUS REPLICATION AND TUMOR GROWTH | VIROSTATICS SRL (IT) | 2011-02-03 | — | — | WO | disclosed |
| US-7666920-B2 | urable molding material an epoxy (meth)acrylate, acrylated polyethers;acrylated bisphenol, and a thermoplastic resin; shape recovering; shape retension; adhesion tosubstrate; high refractive index without a decrease in elastic modulus;Fresnel lens sheet | DAI NIPPON INK AND CHEMICALS, INC. (JP) | 2010-02-23 | — | — | US | disclosed |
| CN-101591281-A | Phosphonate compounds having immunomodulatory activity | GILEAD SCIENCES INC (US) | 2009-12-02 | — | — | CN | disclosed |
| US-20090247488-A1 | ANTI-INFLAMMATORY PHOSPHONATE COMPOUNDS | CANNIZZARO CARINA | 2009-10-01 | — | — | US | disclosed |
| US-7589086-B2 | Substituted pyrazolo[3,4-D]pyrimidines as anti-tumor agents | UNIVERSITA DEGLI STUDI DI SIENA (IT) | 2009-09-15 | — | — | US | disclosed |
| US-20090227543-A1 | PHOSPHONATE COMPOUNDS HAVING IMMUNO-MODULATORY ACTIVITY | CANNIZZARO CARINA | 2009-09-10 | — | — | US | disclosed |
| CN-101475504-A | 2-acetyl-3-amino-3-aryl-acrylic acid esters and preparation thereof | UNIV SOOCHOW (CN) | 2009-07-08 | — | — | CN | disclosed |
| CN-101410120-A | Anti-inflammatory phosphonate compounds | GILEAD SCIENCES INC (US) | 2009-04-15 | — | — | CN | disclosed |
| US-20090069301-A1 | Acridine and Quinoline Derivatives as Sirtuin Modulators | SIRTRIS PHARMACEUTICALS, INC. (US) | 2009-03-12 | — | — | US | disclosed |
| US-7470724-B2 | Phosphonate compounds having immuno-modulatory activity | GILEAD SCIENCES, INC. (US) | 2008-12-30 | — | — | US | disclosed |
| US-7432261-B2 | Anti-inflammatory phosphonate compounds | GILEAD SCIENCES, INC. (US) | 2008-10-07 | — | — | US | disclosed |
| US-20080194590-A1 | 4-Piperazinylthieno [2,3-D] Pyrimidine Compounds as Platelet Aggregation Inhibitors | PFIZER INC | 2008-08-14 | — | — | US | disclosed |
| CN-101218203-A | Derivatives of 4-(2-amino-1-hydroxyethyl) phenol as agonists of the ss2 adrenergic receptor | ALMIRALL PRODESFARMA SA (ES) | 2008-07-09 | — | — | CN | disclosed |
| EP-1638966-B1 | 4-SUBSTITUTED DERIVATIVES OF PYRAZOLO ¬3,4-d PYRIMIDINE AND USES THEREOF | UNIV SIENA (IT) | 2008-03-19 | — | — | EP | disclosed |
| EP-1869051-A1 | 4-PIPERAZINYLTHIENO Ý2,3-D¨PYRIMIDINE COMPOUNDS AS PLATELET AGGREGATION INHIBITORS | Pharmacia & Upjohn Company LLC (US) | 2007-12-26 | — | — | EP | disclosed |
| EP-1856099-A2 | ACRIDINE AND QUINOLINE DERIVATIVES AS SIRTUIN MODULATORS | Sirtris Pharmaceuticals, Inc. (US) | 2007-11-21 | — | — | EP | disclosed |
| CN-101037425-A | 2-furoyl-3-aryl-4-ethoxy acetyl-5-methyl-trans-2,3-Dihydrofuran and preparation method thereof | UNIV SHANGHAI (CN) | 2007-09-19 | — | — | CN | disclosed |
| US-20070010510-A1 | 4-Substituted derivatives of pyrazolo[3,4-d]pyrimidine and pyrrolo[2,3-d]pyrimidine and uses thereof | UNIVERSITA DEGLI STUDI DI SIENA (IT) | 2007-01-11 | — | — | US | disclosed |
| WO-2006103545-A1 | 4-PIPERAZINYLTHIENO [2,3-D] PYRIMIDINE COMPOUNDS AS PLATELET AGGREGATION INHIBITORS | PHARMACIA & UPJOHN COMPANY LLC (US) | 2006-10-05 | — | — | WO | disclosed |
| WO-2006094237-A2 | ACRIDINE AND QUINOLINE DERVATIVES AS SIRTUIN MODULATORS | SIRTRIS PHARMACEUTICALS, INC. (US) | 2006-09-08 | — | — | WO | disclosed |
| US-20060199788-A1 | Anti-inflammatory phosphonate compounds | GILEAD SCIENCES, INC. | 2006-09-07 | — | — | US | disclosed |
| US-20060189706-A1 | Actinic-energy-ray-curable resin composition for lens sheet and lens sheet | DAI NIPPON PRINTING CO., LTD. (JP) | 2006-08-24 | — | — | US | disclosed |
| EP-1663254-A2 | ANTI-INFLAMATORY PHOSPHONATE CONJUGATES | GILEAD SCIENCES, INC. (US) | 2006-06-07 | — | — | EP | disclosed |
| CN-1780630-A | Phosphonate compounds having immunomodulatory activity | GILEAD SCIENCES INC (US) | 2006-05-31 | — | — | CN | disclosed |
| CN-1250644-C | Active energy ray-curable resin composition for Fresnel lens and Fresnel lens sheet | DAINIPPON INK & CHEMICALS (JP) | 2006-04-12 | — | — | CN | disclosed |
| EP-1638966-A2 | 4-SUBSTITUTED DERIVATIVES OF PYRAZOLO ¬3,4-d| PYRIMIDINE AND PYRROLO ¬2,3-d| PYRIMIDINE AND USES THEREOF | UNIVERSITA DEGLI STUDI DI SIENA (IT) | 2006-03-29 | — | — | EP | disclosed |
| US-20060035866-A1 | Phosphonate compounds having immuno-modulatory activity | GILEAD SCIENCES, INC. | 2006-02-16 | — | — | US | disclosed |
| EP-1620110-A2 | IMMUNOMODULATOR PHOSPHONATE CONJUGATES | GILEAD SCIENCES, INC. (US) | 2006-02-01 | — | — | EP | disclosed |
| EP-1308471-B1 | Radiation curable resin composition for Fresnel lens and Fresnel lens sheet | DAINIPPON INK & CHEMICALS (JP) | 2005-12-14 | — | — | EP | disclosed |
| US-6852718-B2 | Phenylsulphonylipiperazinyl derivatives as 5-HT receptor ligands | MERCK SHARP & DOHME LTD | 2005-02-08 | — | — | US | disclosed |
| WO-2004106340-A2 | 4-SUBSTITUTED DERIVATIVES OF PYRAZOLO [3,4-d] PYRIMIDINE AND PYRROLO [2,3-d] PYRIMIDINE AND USES THEREOF | UNIVERSITÀ DEGLI STUDI DI SIENA (IT) | 2004-12-09 | — | — | WO | disclosed |
| WO-2004100960-A2 | ANTI-INFLAMMATORY PHOSPHONATE COMPOUNDS | GILEAD SCIENCES, INC. (US) | 2004-11-25 | — | — | WO | disclosed |
| WO-2004096236-A2 | IMMUNOMODULATOR PHOSPHONATE CONJUGATES | GILEAD SCIENCES, INC. (US) | 2004-11-11 | — | — | WO | disclosed |
| US-6809889-B2 | EPOXY (METH)ACRYLATE; (METH)ACRYLATE OF LOW MOLECULAR WEIGHT POLYOXYPROPYLENE; CYCLIC (METH)ACRYLATE (E.G., PHENOXYETHYL ACRYLATE) AND (METH)ACRYLATE OF TRIS(HYDROXYALKYL) ISOCYANURATE; HIGH ELASTIC MODULUS AND REFRACTIVE INDEX | DAINIPPON INK AND CHEMICALS, INC. (JP) | 2004-10-26 | — | — | US | disclosed |
| CN-1168709-C | Alpha-hydroxy, amino and -fluoro derivatives of beta-sulphenyl hydroxamic acids matrix metalloproteinases inhibitors | ����Լ��ҩ�﹫˾ | 2004-09-29 | — | — | CN | disclosed |
| US-6777430-B2 | A DERIVATIVES WITH ATTACHED TO AN N-ARYLALKYL-SUBSTITUTED AZETIDINE, PYRROLIDINE OR PIPERIDINE RING; A SERATONIN RECEPTOR ANTAGONISTS FOR TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDER SCHIZOPHRENIA, DEPRESSION | MERCK SHARP & DOHME LTD. | 2004-08-17 | — | — | US | disclosed |
| EP-1147084-B1 | PHENYLSULPHONYL DERIVATIVES AS 5-HT RECEPTOR LIGANDS | MERCK SHARP & DOHME (GB) | 2004-05-19 | — | — | EP | disclosed |
| US-20030203889-A1 | Phenylsulphonyl derivatives as 5-HT receptor ligands | MERCK & CO., INC. | 2003-10-30 | — | — | US | disclosed |
| US-20030181464-A1 | Phenylsulphonylipiperazinyl derivatives as 5-ht receptor ligands | THE INSTITUTE OF CANCER RESEARCH (GB) | 2003-09-25 | — | — | US | disclosed |
| US-20030166687-A1 | ALPHA-HYDROXY,-AMINO AND -FLUORO DERIVATIVES OF BETA-SULPHONYL HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASES INHIBITORS | PHARMACIA & UPJOHN COMPANY | 2003-09-04 | — | — | US | disclosed |
| US-20030113544-A1 | Radiation curable resin composition for fresnel lens and fresnel lens sheet | DAINIPPON INK AND CHEMICALS, INC. (JP) | 2003-06-19 | — | — | US | disclosed |
| EP-1308471-A2 | Radiation curable resin composition for Fresnel lens and Fresnel lens sheet | DAINIPPON INK AND CHEMICALS, INC. (JP) | 2003-05-07 | — | — | EP | disclosed |
| US-6559166-B1 | A class of phenylsulphonyl derivatives wherein the sulphonyl moiety is also attached to an N-arylalkyl-substituted azetidine, pyrrolidine or piperidine ring are selective antagonists of the human 5-HT2A receptor and are therefore | MERCK SHARP & DOHME LTD. | 2003-05-06 | — | — | US | disclosed |
| CN-1414030-A | Active energy ray-curable resin composition for Fresnel lens and Fresnel lens sheet | DAINIPPON INK & CHEMICALS (JP) | 2003-04-30 | — | — | CN | disclosed |
| EP-1280785-A1 | PHENYLSULPHONYLPIPERAZINYL DERIVATIVES AS 5-HT RECEPTOR LIGANDS | MERCK SHARP & DOHME LTD. (GB) | 2003-02-05 | — | — | EP | disclosed |
| EP-1037868-B1 | $g(a)-HYDROXY, -AMINO, AND HALO DERIVATIVES OF $g(b)-SULFONYL HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASES INHIBITORS | UPJOHN CO (US) | 2003-02-05 | — | — | EP | disclosed |
| US-6437177-B1 | DISEASES INVOLVING CONNECTIVE TISSUE DEGRADATION; ARTHRITIS, OSTEOPOROSIS, PERIODONTITIS, GINGIVITIS, CORNEAL, DERMAL, OR GASTRIC ULCERATION, AND ASTHMA; 2-HYDROXY-2-(PHENYLTHIO) METHYL-3-(4-BUTOXYBENZENESULFONYL)PROPIONIC ACID | PHARMACIA & UPJOHN COMPANY | 2002-08-20 | — | — | US | disclosed |
| US-6316468-B1 | Phenylindole derivatives as 5-HT2A receptor antagonists | MERCK SHARP & DOHME LTD. | 2001-11-13 | — | — | US | disclosed |
| EP-1147084-A1 | PHENYLSULPHONYL DERIVATIVES AS 5-HT RECEPTOR LIGANDS | MERCK SHARP & DOHME LTD. (GB) | 2001-10-24 | — | — | EP | disclosed |
| WO-2001074797-A1 | PHENYLSULPHONYLPIPERAZINYL DERIVATIVES AS 5-HT RECEPTOR LIGANDS | MERCK SHARP & DOHME LIMITED (GB) | 2001-10-11 | — | — | WO | disclosed |
| US-6235928-B1 | ENZYME INHIBITOR MATRIX METALLOPROTEINASE FAMILY, INCLUDING COLLAGENASE, STROMELYSIN, AND GELATINASE, THE COMPOUNDS OR PHARMACEUTICAL COMPOSITIONS | PHARMACIA & UPJOHN COMPANY | 2001-05-22 | — | — | US | disclosed |
| CN-1278247-A | Alpha-hydroxy, -amino and halo derivatives of beta-sulfonyl hydroxamic acids as matrix metalloproteinase inhibitors | PHARMACIA & UPJHN CO (US) | 2000-12-27 | — | — | CN | disclosed |
| EP-1037868-A2 | $g(a)-HYDROXY, -AMINO, AND HALO DERIVATIVES OF $g(b)-SULFONYL HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASES INHIBITORS | PHARMACIA & UPJOHN COMPANY (US) | 2000-09-27 | — | — | EP | disclosed |
| WO-2000043362-A1 | PHENYLSULPHONYL DERIVATIVES AS 5-HT RECEPTOR LIGANDS | MERCK SHARP & DOHME LIMITED (GB) | 2000-07-27 | — | — | WO | disclosed |
| EP-1002004-A1 | SILICONIMIDES CONTAINING Si-H GROUPS | Wacker-Chemie GmbH (DE) | 2000-05-24 | — | — | EP | disclosed |
| EP-0929519-A1 | $g(b)-SULFONYL HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASES INHIBITORS | PHARMACIA & UPJOHN COMPANY (US) | 1999-07-21 | — | — | EP | disclosed |
| WO-1999026909-A2 | ALPHA-HYDROXY, -AMINO AND -FLUORO DERIVATIVES OF BETA-SULPHONYL HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASES INHIBITORS | PHARMACIA & UPJOHN COMPANY (US) | 1999-06-03 | — | — | WO | disclosed |
| WO-1999011641-A1 | PHENYLINDOLE DERIVATIVES AS 5-HT2A RECEPTOR ANTAGONISTS | MERCK SHARP & DOHME LIMITED (GB) | 1999-03-11 | — | — | WO | disclosed |
| WO-1999007767-A1 | SILICONIMIDES CONTAINING Si-H GROUPS | WACKER-CHEMIE GMBH (DE) | 1999-02-18 | — | — | WO | disclosed |
| US-5847153-A | β-sulfonyl hydroxamic acids | PHARMACIA & UPJOHN COMPANY (US) | 1998-12-08 | — | — | US | disclosed |
| WO-1998013340-A1 | β-SULFONYL HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASES INHIBITORS | PHARMACIA & UPJOHN COMPANY (US) | 1998-04-02 | — | — | WO | disclosed |
| CN-1120313-A | Heart failure remedy | NISSAN CHEMICAL IND LTD (JP) | 1996-04-10 | — | — | CN | disclosed |
| EP-0354788-B1 | Novel imidazole derivatives | NIPPON CHEMIPHAR CO (JP) | 1995-09-13 | — | — | EP | disclosed |
| US-5306719-A | Cardiotonic agents | OTSUKA PHARMACEUTICAL CO., LTD. (JP) | 1994-04-26 | — | — | US | disclosed |
| US-5286395-A | Oil additive | INSTITUT FRANCAIS DU PETROLE (FR) | 1994-02-15 | — | — | US | disclosed |
| EP-0255134-B1 | CARBOSTYRIL DERIVATIVES AND SALTS THEREOF, PROCESS FOR PREPARING THEM, AND CARDIOTONIC COMPOSITION CONTAINING SAME | OTSUKA PHARMACEUTICAL CO., LTD. (JP) | 1993-03-03 | — | — | EP | disclosed |
| US-5180836-A | Antiulcer agents | NIPPON CHEMIPHAR CO., LTD. (JP) | 1993-01-19 | — | — | US | disclosed |
| US-5132031-A | Antiwear Agents, Antioxidants | INSTITUT FRANCAIS DU PETROLE (FR) | 1992-07-21 | — | — | US | disclosed |
| US-5082943-A | Antiulcer | NIPPON CHEMIPHAR CO., LTD. (JP) | 1992-01-21 | — | — | US | disclosed |
| US-5071856-A | CARBOSTYRIL DERIVATIVES AND SALTS THEREOF | OTSUKA PHARMACEUTICAL CO., LTD. (JP) | 1991-12-10 | — | — | US | disclosed |
| US-5045221-A | corrosion resistance; additive to extreme pressure, temperature lubricants | ISTITUT FRANCAIS DU PETROLE (FR) | 1991-09-03 | — | — | US | disclosed |
| EP-0360633-A1 | Polysulphurised olefin composition, its preparation and its use as an additive in lubricants | Institut Français du Pétrole (FR) | 1990-03-28 | — | — | EP | disclosed |
| EP-0354788-A1 | Novel imidazole derivatives | NIPPON CHEMIPHAR CO., LTD. (JP) | 1990-02-14 | — | — | EP | disclosed |
| US-4886809-A | CARDIOTONIC AGENTS | OTSUKA PHARMACEUTICAL CO., LTD. (JP) | 1989-12-12 | — | — | US | disclosed |
| US-4882446-A | MOLYBDENUM COMPLEXES; EXTREME PRESSURE LUBRICANTS; EFFICIENT WEAR RESISTANCE | INSTITUT FRANCAIS DU PETROLE (FR) | 1989-11-21 | — | — | US | disclosed |
| US-4766228-A | Metal dihydrocarbyl-dithiophosphyl-dithiophosphates their manufacture and use as additives for lubricants | INSTITUT FRANCAIS DU PETROLE (FR) | 1988-08-23 | — | — | US | disclosed |
| EP-0255134-A2 | Carbostyril derivatives and salts thereof, process for preparing them, and cardiotonic composition containing same | OTSUKA PHARMACEUTICAL CO., LTD. (JP) | 1988-02-03 | — | — | EP | disclosed |
| US-4645610-A | EXTREME PRESSURE LUBRICANTS; TRANSMISSION FLUIDS; CUTTING OILS | INSTITUT FRANCAIS DU PETROLE (FR) | 1987-02-24 | — | — | US | disclosed |
| US-4235779-A | Bicyclic lactones | THE UPJOHN COMPANY (US) | 1980-11-25 | — | — | US | disclosed |
| US-4111933-A | PROTECTION OF FUNCTIONAL GROUPS DURING REACTION AND THEIR SUBSEQUENT RESTORATION | BAYER AKTIENGESELLSCHAFT (DE) | 1978-09-05 | — | — | US | disclosed |
| US-4111933-A | PROTECTION OF FUNCTIONAL GROUPS DURING REACTION AND THEIR SUBSEQUENT RESTORATION | BAYER AKTIENGESELLSCHAFT (DE) | 1978-09-05 | — | — | US | disclosed |