SCHEMBL4183465

SCHEMBL4183465

Cc1ccc(C(=O)N2CCC(c3ccc(C(=O)N(C)C)cc3)CC2)cc1NS(=O)(=O)Cc1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FASN P49327 14/20 0.45
CCR1 P32246 1/20 0.45
KMT2A Q03164 2/20 0.44
HDAC1 Q13547 1/20 0.43
MEN1 O00255 1/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
CYP3A4 P08684 1/20 0.43
GAA P10253 1/20 0.43
HPGD P15428 1/20 0.43
CYP2C19 P33261 1/20 0.43
HTT P42858 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA7 P43166 1/20 0.42
CA9 Q16790 1/20 0.42
CA14 Q9ULX7 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4786009 0.90 FASN (0.51) FASN
SCHEMBL4172391 0.89 CA12 (0.48) FASNCCR1KMT2AMEN1ALDH1A1
SCHEMBL31615499 0.88 PARP10 (0.52) FASNCCR1KMT2AHTT
SCHEMBL4176902 0.88 FASN (0.59) FASN
SCHEMBL4187269 0.85 FASN (0.57) FASN
SCHEMBL31615859 0.85 FASN (0.46) FASNCCR1
SCHEMBL31615826 0.84 FASN (0.45) FASNCCR1KMT2AMEN1ALDH1A1
SCHEMBL31615805 0.83 PARP14 (0.45) FASNCCR1
SCHEMBL31615627 0.83 PARP10 (0.45) FASNCCR1CYP3A4GAACYP2C19
Methanesulfonamide SCHEMBL4737271 0.83 FASN (0.54) FASNCA12CA1CA2CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090105305-A1 Therapeutic Agents - 550 ASTRAZENECA AB (SE) 2009-04-23 US disclosed
WO-2008075070-A1 SULFONAMIDE DERIVATIVES FOR THERAPEUTIC USE AS FATTY ACID SYNTHASE INHIBITORS ASTRAZENECA AB (SE) 2008-06-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090105305-A1 Therapeutic Agents - 550 FABP4, GPR119, FASN FASN 3/4885CCR1 1814/4885KMT2A 3544/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.