SCHEMBL4184375

SCHEMBL4184375

FC(F)(F)c1ccnc(Nc2cccc(Cl)c2)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 3/20 0.55
HTR3E A5X5Y0 1/20 0.54
HTR3B O95264 1/20 0.54
HTR3A P46098 1/20 0.54
ROCK1 Q13464 1/20 0.54
HTR3D Q70Z44 1/20 0.54
HTR3C Q8WXA8 1/20 0.54
THRB P10828 1/20 0.51
FADS1 O60427 2/20 0.51
MEN1 O00255 1/20 0.50
ALDH1A1 P00352 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
MAPT P10636 1/20 0.50
CYP2C19 P33261 1/20 0.50
KMT2A Q03164 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
KIF11 P52732 4/20 0.48
EGFR P00533 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3956336 0.80 HTR3E (0.57) HTR3EHTR3BHTR3AROCK1HTR3D
SCHEMBL4238979 0.80 AURKA (0.67) AURKATHRBMEN1ALDH1A1CYP1A2
SCHEMBL1518750 0.79 AURKA (0.65) AURKATHRBMAPTKIF11EGFR
SCHEMBL3206970 0.78 AURKA (0.70) AURKAHTR3EHTR3BHTR3AROCK1
SCHEMBL20172492 0.78 KIF11 (0.66) AURKATHRBMEN1KMT2AKIF11
SCHEMBL3951446 0.77 HTR3E (0.57) HTR3EHTR3BHTR3AROCK1HTR3D
SCHEMBL30643204 0.77 GRM5 (0.62) AURKAMEN1ALDH1A1MAPTKMT2A
SCHEMBL30847438 0.77 AURKA (0.62) AURKATHRBMEN1ALDH1A1CYP1A2
SCHEMBL27112491 0.77 AURKA (0.62) AURKATHRBMEN1ALDH1A1CYP1A2
SCHEMBL4737841 0.76 GAK (0.69) FADS1EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009029617-A1 DIARYLAMINE-SUBSTITUTED QUINOLONES USEFUL AS INDUCIBLE NITRIC OXIDE SYNTHASE INHIBITORS KALYPSYS, INC. (US) 2009-03-05 WO disclosed