SCHEMBL4184590

SCHEMBL4184590

Cc1nc(NC(=O)c2ccccc2C(F)(F)F)sc1C(=O)O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 10/20 0.58
NPC1 O15118 8/20 0.58
SMN1; SMN2 Q16637 5/20 0.58
PKM P14618 4/20 0.58
TP53 P04637 1/20 0.58
ALOX15 P16050 1/20 0.58
HTT P42858 1/20 0.58
HSD17B10 Q99714 1/20 0.58
ALDH1A1 P00352 4/20 0.57
TDP1 Q9NUW8 1/20 0.55
NPSR1 Q6W5P4 2/20 0.54
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
RXFP1 Q9HBX9 1/20 0.50
PDE5A O76074 1/20 0.49
PDE1A P54750 1/20 0.49
PDE1B Q01064 1/20 0.49
PDE1C Q14123 1/20 0.49
HPGD P15428 2/20 0.49
KDM4E B2RXH2 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3586382 0.86 SCD (0.65) RAB9ANPC1SMN1; SMN2PKMTP53
SCHEMBL28773907 0.85 PKM (0.46) RAB9ANPC1SMN1; SMN2PKMTP53
SCHEMBL3585640 0.84 RAB9A (0.81) RAB9ANPC1SMN1; SMN2PKMTP53
SCHEMBL3584894 0.83 RAB9A (0.80) RAB9ANPC1SMN1; SMN2PKMTP53
SCHEMBL4338019 0.82 RAB9A (0.57) RAB9ANPC1SMN1; SMN2PKMTP53
SCHEMBL4196428 0.80 SMN1; SMN2 (0.81) RAB9ANPC1SMN1; SMN2PKMTP53
SCHEMBL3582729 0.79 NPC1 (0.73) RAB9ANPC1SMN1; SMN2PKMTP53
SCHEMBL4199061 0.79 NPC1 (0.63) RAB9ANPC1SMN1; SMN2PKMHTT
SCHEMBL4195858 0.78 RAB9A (0.57) RAB9ANPC1SMN1; SMN2PKMTP53
SCHEMBL3584043 0.77 RAB9A (0.81) RAB9ANPC1SMN1; SMN2PKMTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029138-A1 AMINOTHIAZOLE DERIVATIVES AS HUMAN STEAROYL-COA DESATURASE INHIBITORS XENON PHARMACEUTICALS INC. (CA) 2009-03-04 EP disclosed
WO-2007130075-A1 AMINOTHIAZOLE DERIVATIVES AS HUMAN STEAROYL-COA DESATURASE INHIBITORS XENON PHARMACEUTICALS INC. (CA) 2007-11-15 WO disclosed