SCHEMBL4187153

SCHEMBL4187153

Cc1ccc(S(=O)(=O)Cl)c(O)c1C

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 2/20 0.35
ALDH1A1 P00352 7/20 0.35
POLB P06746 1/20 0.35
RECQL P46063 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
TDP2 O95551 1/20 0.34
NSD2 O96028 1/20 0.34
HSP90AA1 P07900 1/20 0.34
PAX8 Q06710 1/20 0.34
GAA P10253 4/20 0.34
TSHR P16473 3/20 0.34
HSD17B10 Q99714 2/20 0.34
ALOX15 P16050 1/20 0.34
KMT2A Q03164 3/20 0.33
PKM P14618 2/20 0.33
MEN1 O00255 2/20 0.33
LMNA P02545 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4758230 0.82 TRPV4 (0.38) TRPV4ALDH1A1GAATSHRHSD17B10
SCHEMBL2227316 0.81 MEN1 (0.41) ALDH1A1POLBRECQLNPSR1TDP1
SCHEMBL30039434 0.80 ALDH1A1 (0.44) TRPV4ALDH1A1POLBTDP1TDP2
SCHEMBL2930464 0.80 ALDH1A1 (0.44) TRPV4ALDH1A1POLBTDP1TDP2
SCHEMBL216318 0.75 ALDH1A1 (0.52) ALDH1A1TDP1GAATSHRHSD17B10
SCHEMBL31453875 0.72 TRPV4 (0.40) TRPV4ALDH1A1NPSR1TDP2NSD2
SCHEMBL2266737 0.72 TRPV4 (0.36) TRPV4ALDH1A1TDP1TDP2NSD2
SCHEMBL4618011 0.71 KMT2A (0.39) TRPV4ALDH1A1TDP2NSD2HSP90AA1
SCHEMBL29907244 0.71 TRPV4 (0.35) TRPV4ALDH1A1TDP2NSD2HSP90AA1
SCHEMBL907691 0.71 GAA (0.50) ALDH1A1POLBRECQLTDP1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090069302-A1 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2009-03-12 US disclosed
EP-1976498-A2 CHEMICAL COMPOUNDS SmithKline Beecham Corporation (US) 2008-10-08 EP disclosed
WO-2007127505-A2 USE OF SULFONAMIDE DERIVATIVES IN THE TREATMENT OF DISORDERS OF THE METABOLISM AND THE NERVOUS SYSTEM SMITHKLINE BEECHAM CORPORATION (US) 2007-11-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090069302-A1 CHEMICAL COMPOUNDS TBXA2R, PDE4D, PDE4A TRPV4 54/4885ALDH1A1 669/4885POLB 4819/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.