SCHEMBL4187652

SCHEMBL4187652

COC(=O)c1sc2ccccc2c1NC(=O)CCSc1ccc(Br)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.49
L3MBTL1 Q9Y468 3/20 0.49
KDM4E B2RXH2 2/20 0.49
HSD17B10 Q99714 2/20 0.49
TSHR P16473 1/20 0.49
LMNA P02545 4/20 0.45
MAPK1 P28482 1/20 0.45
MEN1 O00255 2/20 0.45
MAPT P10636 2/20 0.45
KMT2A Q03164 2/20 0.45
POLB P06746 1/20 0.45
PKM P14618 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
TP53 P04637 1/20 0.45
GLA P06280 1/20 0.44
GAA P10253 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4181297 0.91 ALDH1A1 (0.53) ALDH1A1L3MBTL1KDM4EHSD17B10TSHR
SCHEMBL4185817 0.89 ALDH1A1 (0.51) ALDH1A1L3MBTL1KDM4EHSD17B10TSHR
SCHEMBL4196894 0.80 ALDH1A1 (0.55) ALDH1A1L3MBTL1KDM4EHSD17B10TSHR
SCHEMBL31538574 0.78 ALDH1A1 (0.60) ALDH1A1L3MBTL1KDM4EHSD17B10TSHR
SCHEMBL4333252 0.78 ALDH1A1 (0.60) ALDH1A1L3MBTL1KDM4EHSD17B10TSHR
SCHEMBL4194030 0.77 LMNA (0.55) ALDH1A1KDM4EHSD17B10TSHRLMNA
SCHEMBL4187568 0.76 ALDH1A1 (0.47) ALDH1A1L3MBTL1KDM4EHSD17B10TSHR
SCHEMBL4751448 0.75 KMT2A (0.65) ALDH1A1L3MBTL1LMNAMEN1MAPT
SCHEMBL4734529 0.74 KDM4E (0.64) ALDH1A1L3MBTL1KDM4ELMNAMEN1
SCHEMBL4178799 0.73 NPSR1 (0.47) ALDH1A1KDM4EKMT2ACYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009048274-A2 BENZOFURAN AND BENZOTHIOPHENE DERIVATIVES SUBSTITUTED WITH AMIDE, PROCESS FOR THE PREPARATION THEREOF, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2009-04-16 WO claimed
WO-2009048274-A2 BENZOFURAN AND BENZOTHIOPHENE DERIVATIVES SUBSTITUTED WITH AMIDE, PROCESS FOR THE PREPARATION THEREOF, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2009-04-16 WO disclosed