SCHEMBL4188079

SCHEMBL4188079

C#Cc1ccc(CC(NC(=O)c2c(C)cc(C)cc2C)C(=O)O)cc1

nearest known ligand 0.64

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 18/20 0.64
ITGA4 P13612 4/20 0.64
L3MBTL1 Q9Y468 1/20 0.57
ITGB3 P05106 14/20 0.57
ITGAV P06756 14/20 0.57
ITGA5 P08648 14/20 0.57
ITGA2B P08514 12/20 0.57
ITGB5 P18084 10/20 0.50
ITGA2 P17301 1/20 0.49
ITGB7 P26010 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16378072 0.85 ITGB1 (0.66) ITGB1ITGA4L3MBTL1ITGB3ITGAV
SCHEMBL4170016 0.84 L3MBTL1 (0.79) ITGB1ITGA4L3MBTL1ITGB3ITGAV
SCHEMBL4513437 0.84 ITGB1 (0.50) ITGB1ITGA4L3MBTL1ITGB3ITGAV
SCHEMBL8230444 0.84 ITGB1 (0.50) ITGB1ITGA4L3MBTL1ITGB3ITGAV
SCHEMBL4527614 0.81 ITGB1 (0.62) ITGB1ITGA4L3MBTL1ITGB3ITGAV
SCHEMBL6516795 0.77 ITGA4 (0.66) ITGB1ITGA4L3MBTL1ITGB3ITGAV
SCHEMBL4194979 0.76 NLRP3 (0.59) ITGB1ITGA4L3MBTL1ITGB3ITGAV
SCHEMBL8232058 0.76 NLRP3 (0.59) ITGB1ITGA4L3MBTL1ITGB3ITGAV
SCHEMBL13881435 0.76 PPARG (0.43) ITGB1ITGA4L3MBTL1ITGB3ITGA2B
SCHEMBL28965860 0.76 PTPN1 (0.65) L3MBTL1ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2024357-A2 NEW HETEROCYCLIC COMPOUNDS FOR THE INHIBITION OF INTEGRINS AND USE THEREOF Jereni AG (DE) 2009-02-18 EP disclosed
WO-2007131764-A2 NEW HETEROCYCLIC COMPOUNDS FOR THE INHIBITION OF INTEGRINS AND USE THEREOF JERINI AG (DE) 2007-11-22 WO disclosed