SCHEMBL6516795

SCHEMBL6516795

Cc1cc(C)c(C(=O)N[C@@H](Cc2ccc(OCc3c(Cl)cccc3Cl)cc2)C(=O)O)c(C)c1

nearest known ligand 0.66

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 14/20 0.66
ITGB1 P05556 12/20 0.66
ITGA5 P08648 5/20 0.62
ITGB3 P05106 3/20 0.62
ITGAV P06756 3/20 0.62
ITGA2 P17301 1/20 0.54
ITGB7 P26010 1/20 0.54
L3MBTL1 Q9Y468 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6515404 0.84 ITGB1 (0.65) ITGA4ITGB1ITGA5ITGB3ITGAV
SCHEMBL7616517 0.83 ITGA4 (0.54) ITGA4ITGB1ITGA5ITGB3ITGAV
SCHEMBL7612266 0.81 ITGA4 (0.60) ITGA4ITGB1ITGA5ITGB3ITGAV
SCHEMBL3722481 0.81 ITGA4 (0.67) ITGA4ITGB1
SCHEMBL3722480 0.81 ITGA4 (0.67) ITGA4ITGB1
SCHEMBL7608992 0.80 ITGA4 (0.69) ITGA4ITGB1ITGA5ITGB3ITGAV
SCHEMBL7605621 0.80 GPR132 (0.60) ITGA4ITGB1
SCHEMBL7605500 0.80 ITGB1 (0.60) ITGA4ITGB1ITGA5ITGB3ITGAV
SCHEMBL7991610 0.79 ITGA4 (0.53) ITGA4ITGB1ITGA5ITGB3ITGAV
SCHEMBL4170016 0.79 L3MBTL1 (0.79) ITGA4ITGB1ITGA5ITGB3ITGAV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050215598-A1 Phenylalanine derivatives CELLTECH R&D LTD. (GB) 2005-09-29 US disclosed
US-20030166691-A1 Phenylalanine derivatives ARCHIBALD SARAH CATHERINE (GB) 2003-09-04 US disclosed
US-6555562-B1 2-Carboxybenzoyl-(N'-3,5-dichloroisonicotinoyl)-L-4aminophenyl alanine, for example; inhibit the binding of alpha-4 integrins to their ligands, use to treat immune or inflammatory disorders CELLTECH R&D LIMITED (GB) 2003-04-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030166691-A1 Phenylalanine derivatives VCAM1, PAH, ITGB4 ITGA4 4/4885ITGB1 6/4885ITGA5 28/4885
US-20050215598-A1 Phenylalanine derivatives PAH, ITGB4, VCAM1 ITGA4 4/4885ITGB1 7/4885ITGA5 29/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.