SCHEMBL4188375

SCHEMBL4188375

N#Cc1ccc(-c2cccc(C(=O)O)c2C(F)(F)F)cc1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
BRS3 P32247 1/20 0.45
PTGDR2 Q9Y5Y4 1/20 0.43
XDH P47989 5/20 0.43
SLC22A12 Q96S37 5/20 0.43
KIF11 P52732 1/20 0.42
LTB4R2 Q9NPC1 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
TAS2R14 Q9NYV8 1/20 0.41
HNF4A P41235 1/20 0.41
PDK2 Q15119 1/20 0.39
PTPN5 P54829 1/20 0.39
CYP11B2 P19099 1/20 0.39
RXRA P19793 1/20 0.39
RXRG P48443 1/20 0.39
HTT P42858 1/20 0.38
PARP1 P09874 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2174123 0.83 HNF4A (0.58) TAS2R14HNF4A
SCHEMBL2426967 0.81 KAT6A (0.47) BRS3XDHSLC22A12LTB4R2HDAC1
SCHEMBL6164290 0.80 BRS3 (0.57) BRS3XDHSLC22A12LTB4R2HNF4A
SCHEMBL940482 0.79 HSD17B10 (0.48) TAS2R14HNF4A
SCHEMBL11805019 0.79 BRS3 (0.56) BRS3XDHSLC22A12LTB4R2HNF4A
SCHEMBL2744720 0.78 TSHR (0.47) BRS3XDHSLC22A12LTB4R2HNF4A
SCHEMBL2744074 0.78 LTB4R2 (0.46) BRS3XDHSLC22A12LTB4R2HNF4A
SCHEMBL2744830 0.74 LTB4R2 (0.44) BRS3XDHSLC22A12LTB4R2HNF4A
SCHEMBL28481844 0.74 ALDH1A1 (0.52) TAS2R14
SCHEMBL28334899 0.74 DDT (0.54) HDAC1HDAC6HNF4APDK2RXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2021328-A2 COMPOUNDS AND COMPOSITIONS AS HEDGEHOG PATHWAY MODULATORS IRM LLC (BM) 2009-02-11 EP disclosed
WO-2007131201-A2 COMPOUNDS AND COMPOSITIONS AS HEDGEHOG PATHWAY MODULATORS IRM LLC (BM) 2007-11-15 WO disclosed