SCHEMBL4190944

SCHEMBL4190944

Nc1noc2cc(-c3cc(Cl)c(CC4CN(N5CCCC5=O)CCC4O)c(Cl)c3)ccc12

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 1/20 0.33
LCK P06239 1/20 0.31
CSF1R P07333 1/20 0.31
F7 P08709 1/20 0.30
F11 P03951 3/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4191491 0.86 MAPK14 (0.32) MAPK14LCKCSF1R
SCHEMBL1093469 0.77 MAPK14 (0.35) MAPK14LCKCSF1RF7F11
SCHEMBL1093467 0.77 MAPK14 (0.35) MAPK14LCKCSF1RF7F11
SCHEMBL4181628 0.77
SCHEMBL4196923 0.75 HPGD (0.42)
SCHEMBL4185003 0.73 PDE5A (0.34)
SCHEMBL4183670 0.72 SPR (0.34)
SCHEMBL4180585 0.70 S1PR5 (0.40)
SCHEMBL1092474 0.69 MAPK14 (0.31) MAPK14LCKCSF1R
SCHEMBL1092472 0.69 MAPK14 (0.31) MAPK14LCKCSF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2021336-A2 INHIBITORS OF 11-BETA-HYDROXYSTEROID DEHYDROGENASE 1 ELI LILLY AND COMPANY (US) 2009-02-11 EP disclosed
WO-2007127688-A2 INHIBITORS OF 11-BETA-HYDROXYSTEROID DEHYDROGENASE 1 ELI LILLY AND COMPANY (US) 2007-11-08 WO disclosed