SCHEMBL4197311

SCHEMBL4197311

CC(NCC(F)(F)F)(c1cccnc1)c1cccnc1

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.44
L3MBTL1 Q9Y468 1/20 0.43
LMNA P02545 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
KIF11 P52732 2/20 0.40
KCNA5 P22460 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13557773 0.74 CYP19A1 (0.55) CYP19A1LMNACYP1A2CYP3A4CYP11B1
SCHEMBL28036808 0.74 CYP19A1 (0.55) CYP19A1LMNACYP1A2CYP3A4CYP11B1
SCHEMBL10044245 0.72 CYP19A1 (0.49) CYP19A1LMNACYP1A2CYP3A4CYP11B1
SCHEMBL27888098 0.71 CYP19A1 (0.52) CYP19A1LMNACYP1A2CYP3A4CYP11B1
SCHEMBL22303441 0.71 CYP19A1 (0.52) CYP19A1LMNACYP1A2CYP3A4CYP11B1
SCHEMBL10202596 0.70 CYP19A1 (0.47) CYP19A1LMNACYP1A2CYP3A4CYP11B1
SCHEMBL3021832 0.70 CYP19A1 (0.55) CYP19A1LMNACYP1A2CYP3A4CYP11B1
SCHEMBL28276861 0.70 CYP19A1 (0.55) CYP19A1LMNACYP1A2CYP3A4CYP11B1
SCHEMBL31507922 0.70 KCNA5 (0.47) CYP19A1LMNACYP1A2CYP3A4CYP11B1
SCHEMBL74389 0.69 KIF11 (0.61) CYP19A1L3MBTL1LMNACYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1781635-A4 POTASSIUM CHANNEL INHIBITORS MERCK & CO INC (US) 2009-02-25 EP disclosed
EP-1781635-A2 POTASSIUM CHANNEL INHIBITORS Merck & Co., Inc. (US) 2007-05-09 EP disclosed
WO-2006015159-A2 POTASSIUM CHANNEL INHIBITORS MERCK & CO., INC. (US) 2006-02-09 WO disclosed