SCHEMBL4210140

SCHEMBL4210140

CCOC(=O)N1CCC(C(=O)O)CC1

nearest known ligand 0.71

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.71
ALDH1A1 P00352 5/20 0.60
SMN1; SMN2 Q16637 2/20 0.59
CHRM1 P11229 1/20 0.59
NPC1 O15118 1/20 0.59
RAB9A P51151 1/20 0.59
L3MBTL1 Q9Y468 2/20 0.56
THRB P10828 1/20 0.56
ATM Q13315 1/20 0.56
MAPT P10636 4/20 0.55
PKM P14618 1/20 0.55
HTT P42858 2/20 0.54
NOS3 P29474 1/20 0.53
NOS2 P35228 1/20 0.53
TSHR P16473 2/20 0.52
TP53 P04637 1/20 0.51
TDP1 Q9NUW8 1/20 0.51
LMNA P02545 1/20 0.50
POLB P06746 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14810258 0.90 CHRM1 (0.76) GAAALDH1A1SMN1; SMN2CHRM1NPC1
SCHEMBL9214032 0.89 GAA (0.62) GAAALDH1A1SMN1; SMN2CHRM1NPC1
SCHEMBL11578382 0.87 GAA (0.56) GAAALDH1A1SMN1; SMN2CHRM1NPC1
SCHEMBL28118094 0.86 GAA (0.73) GAAALDH1A1SMN1; SMN2CHRM1L3MBTL1
SCHEMBL14964905 0.85 CHRM1 (0.68) GAAALDH1A1SMN1; SMN2CHRM1NPC1
SCHEMBL1720494 0.85 MAPT (0.72) GAAALDH1A1CHRM1L3MBTL1THRB
SCHEMBL12436957 0.85 GAA (0.71) GAAALDH1A1SMN1; SMN2CHRM1L3MBTL1
SCHEMBL355693 0.84 SMN1; SMN2 (0.58) GAAALDH1A1SMN1; SMN2CHRM1NPC1
SCHEMBL3629079 0.84 GAA (0.70) GAAALDH1A1SMN1; SMN2CHRM1L3MBTL1
SCHEMBL3346477 0.83 SMN1; SMN2 (0.58) GAAALDH1A1SMN1; SMN2CHRM1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 30 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103214457-A Azole antifungal compound and preparation method and application thereof UNIV PLA 2ND MILITARY MEDICAL 2013-07-24 CN claimed
US-20250074875-A1 AT2R ANTAGONISTS AND USES THEREOF ELI LILLY AND COMPANY 2025-03-06 US disclosed
US-20250042914-A1 PIKFYVE KINASE INHIBITOR HANMI PHARM. CO., LTD. (KR) 2025-02-06 US disclosed
EP-4410795-A1 PIKFYVE KINASE INHIBITOR Hanmi Pharm. Co., Ltd. (KR) 2024-08-07 EP disclosed
CN-118019744-A PIKfyve kinase inhibitors 韩美药品株式会社 2024-05-10 CN disclosed
US-20240084067-A1 NOVEL CURABLE COMPOSITION CONTAINING CYCLIC MONOMER TOKUYAMA CORPORATION (JP) 2024-03-14 US disclosed
EP-4286435-A1 NOVEL CURABLE COMPOSITION CONTAINING CYCLIC MONOMER Tokuyama Corporation (JP) 2023-12-06 EP disclosed
WO-2023055181-A1 PIKFYVE KINASE INHIBITOR 한미약품 주식회사 2023-04-06 WO disclosed
WO-2022163765-A1 NOVEL CURABLE COMPOSITION CONTAINING CYCLIC MONOMER 株式会社トクヤマ 2022-08-04 WO disclosed
CN-103214457-B Azole antifungal compound and preparation method and application thereof THE SECOND MILITARY MEDICAL UNIVERSITY (CN) 2015-08-26 CN disclosed
US-5663200-A CARBAMOYL PEPTIDE DERIVATIVES AS VIRICIDES CIBA-GEIGY CORPORATION (US) 1997-09-02 US disclosed
EP-0542671-B1 Substituted hydroquinone derivatives as intermediates of benzofuran derivatives CIBA GEIGY AG (CH) 1997-01-02 EP disclosed
EP-0708085-A2 Antiviral ethers of aspartate protease substrate isosteres CIBA-GEIGY AG (CH) 1996-04-24 EP disclosed
CN-1089253-A The hydroquinone derivatives that replaces CIBA GEIGY AG (CH) 1994-07-13 CN disclosed
US-5290939-A Process for the manufacture of brofaromine and analogs thereof CIBA-GEIGY CORPORATION (US) 1994-03-01 US disclosed
EP-0542671-A1 Substituted hydroquinone derivatives as intermediates of benzofuran derivatives CIBA-GEIGY AG (CH) 1993-05-19 EP disclosed
EP-0520336-A2 Aldehyde derivatives and their use as calpain inhibitors FUJIREBIO Inc. (JP) 1992-12-30 EP disclosed
US-4987132-A PLATELET ACTIVATING FACTOR ANTAGONISTS YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1991-01-22 US disclosed
EP-0279681-A2 Saturated heterocyclic carboxamide derivatives YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1988-08-24 EP disclosed
EP-0000167-A1 1,2,3,6-Tetrahydroisonicotinic acid and derivatives thereof, methods and starting products for their preparation, and pharmaceutical compositions containing them. Krogsgaard-Larsen, Povl (DK) 1979-01-10 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250042914-A1 PIKFYVE KINASE INHIBITOR PIKFYVE, PIP4K2B, PIP4K2C GAA 1842/4885ALDH1A1 4861/4885SMN1; SMN2 3220/4885
US-20250074875-A1 AT2R ANTAGONISTS AND USES THEREOF AGTR2, AGTR1, AVPR2 GAA 4330/4885ALDH1A1 1253/4885SMN1; SMN2 3687/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.