SCHEMBL4221971

SCHEMBL4221971

Nc1cccc2c1CCc1ccccc1C2=O

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CES1 P23141 2/20 0.59
MAPK14 Q16539 5/20 0.52
MAPK13 O15264 1/20 0.52
MAPK12 P53778 1/20 0.52
MAPK11 Q15759 1/20 0.52
AKR1B1 P15121 2/20 0.51
TDP1 Q9NUW8 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
PARP1 P09874 1/20 0.49
MAOA P21397 2/20 0.48
ADORA2A P29274 1/20 0.47
MAOB P27338 2/20 0.44
PTPRC P08575 1/20 0.43
DYRK1A Q13627 1/20 0.42
BCHE P06276 1/20 0.41
MIF P14174 1/20 0.40
CYP2A6 P11509 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11673017 0.84 MAOA (0.61) CES1MAPK14MAPK13MAPK12MAPK11
SCHEMBL16559358 0.83 NPC1 (0.47) CES1MAPK14MAPK13MAPK12MAPK11
SCHEMBL11905992 0.83 MAPK14 (0.65) CES1MAPK14MAPK13MAPK12MAPK11
SCHEMBL44496 0.80 CES1 (0.90) CES1MAPK14MAPK13MAPK12MAPK11
SCHEMBL29437756 0.80 CES1 (0.90) CES1MAPK14MAPK13MAPK12MAPK11
SCHEMBL29408351 0.80 CES1 (0.90) CES1MAPK14MAPK13MAPK12MAPK11
SCHEMBL7820829 0.80 CES1 (0.61) CES1MAPK14MAPK13MAPK12MAPK11
SCHEMBL8076308 0.79 CES1 (0.59) CES1MAPK14AKR1B1TDP1L3MBTL1
SCHEMBL9642938 0.79 CES1 (0.59) CES1MAPK14AKR1B1TDP1L3MBTL1
SCHEMBL4175611 0.79 CES1 (0.59) CES1MAPK14AKR1B1TDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090105327-A1 Dibenzocycloheptane compounds and pharmaceuticals containing these compounds MERCKLE GMBH (DE) 2009-04-23 US disclosed
EP-1881968-A2 DIBENZOCYCLOHEPTANE COMPOUNDS AND PHARMACEUTICALS CONTAINING THESE COMPOUNDS MERCKLE GMBH (DE) 2008-01-30 EP disclosed
WO-2006120010-A2 DIBENZOCYCLOHEPTANE COMPOUNDS AND PHARMACEUTICALS CONTAINING THESE COMPOUNDS MERCKLE GMBH (DE) 2006-11-16 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090105327-A1 Dibenzocycloheptane compounds and pharmaceuticals containing these compounds BDKRB1, IL1R1, IL1A CES1 156/4885MAPK14 3479/4885MAPK13 3037/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.