SCHEMBL8076308

SCHEMBL8076308

O=C1c2ccccc2CCc2c(Br)cccc21

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 2/20 0.59
TDP1 Q9NUW8 1/20 0.57
L3MBTL1 Q9Y468 1/20 0.57
AKR1B1 P15121 2/20 0.51
PARP10 Q53GL7 1/20 0.49
PARP11 Q9NR21 1/20 0.49
MAOA P21397 2/20 0.48
MAOB P27338 3/20 0.44
PIM1 P11309 1/20 0.43
CSNK1A1 P48729 1/20 0.43
CDK5 Q00535 1/20 0.43
ROCK1 Q13464 1/20 0.43
DYRK1A Q13627 1/20 0.43
LRRK2 Q5S007 1/20 0.43
CLK4 Q9HAZ1 1/20 0.43
DYRK1B Q9Y463 1/20 0.43
BCHE P06276 1/20 0.41
MAPK14 Q16539 1/20 0.41
MIF P14174 3/20 0.40
CYP2A6 P11509 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7052870 0.89 PARP10 (0.58) CES1TDP1L3MBTL1AKR1B1PARP10
SCHEMBL27537662 0.85 PARP10 (0.46) CES1TDP1L3MBTL1PARP10PARP11
SCHEMBL28322695 0.84 MAOA (0.61) CES1TDP1L3MBTL1AKR1B1PARP10
SCHEMBL7054532 0.83 TDP1 (0.69) CES1TDP1L3MBTL1AKR1B1PARP10
SCHEMBL7055100 0.83 CES1 (0.60) CES1TDP1L3MBTL1AKR1B1MAOA
SCHEMBL16163913 0.81 TDP1 (0.66) CES1TDP1L3MBTL1AKR1B1MAOA
SCHEMBL44496 0.80 CES1 (0.90) CES1TDP1L3MBTL1AKR1B1PARP10
SCHEMBL29408351 0.80 CES1 (0.90) CES1TDP1L3MBTL1AKR1B1PARP10
SCHEMBL29437756 0.80 CES1 (0.90) CES1TDP1L3MBTL1AKR1B1PARP10
SCHEMBL28158777 0.80 PARP10 (0.42) CES1TDP1L3MBTL1PARP10PARP11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1042268-A1 DIBENZOSUBERONE DERIVATIVES AND PROCEDURES FOR THEIR PREPARATION Belupo - Lijekovi I Kozmetika D.O.O. (HR) 2000-10-11 EP claimed
WO-1999028284-A1 DIBENZOSUBERONE DERIVATIVES AND PROCEDURES FOR THEIR PREPARATION BELUPO - LIJEKOVI I KOZMETIKA D.O.O. (HR) 1999-06-10 WO claimed
EP-1042268-A1 DIBENZOSUBERONE DERIVATIVES AND PROCEDURES FOR THEIR PREPARATION Belupo - Lijekovi I Kozmetika D.O.O. (HR) 2000-10-11 EP disclosed
WO-1999028284-A1 DIBENZOSUBERONE DERIVATIVES AND PROCEDURES FOR THEIR PREPARATION BELUPO - LIJEKOVI I KOZMETIKA D.O.O. (HR) 1999-06-10 WO disclosed
US-4003915-A ANTICONVULSANTS, PARKINSON*S DISEASE HOFFMANN-LA ROCHE INC. (US) 1977-01-18 US disclosed