SCHEMBL422347

SCHEMBL422347

Cc1cncc2ccccc12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 5/20 0.52
ALDH1A1 P00352 3/20 0.52
CYP1A2 P05177 5/20 0.46
PRKCZ Q05513 1/20 0.46
CYP11B2 P19099 6/20 0.45
CYP11B1 P15538 4/20 0.45
ADRA2A P08913 1/20 0.44
ADRA2B P18089 1/20 0.44
ADRA2C P18825 1/20 0.44
ADRA1A P35348 1/20 0.44
TSHR P16473 2/20 0.43
KDM4E B2RXH2 1/20 0.41
GPR3 P46089 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2B6 P20813 1/20 0.41
CYP2C19 P33261 1/20 0.41
MAPT P10636 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL30901629 0.98 CYP2A6 (0.50) CYP2A6ALDH1A1CYP1A2PRKCZCYP11B2
Ammonia Solution, Strong SCHEMBL28546873 0.98 CYP2A6 (0.50) CYP2A6ALDH1A1CYP1A2PRKCZCYP11B2
SCHEMBL24622042 0.80 CYP1A2 (0.42) CYP2A6ALDH1A1CYP1A2CYP11B2CYP11B1
SCHEMBL21803768 0.79 HPRT1 (0.50) CYP2A6ALDH1A1CYP1A2TSHRCYP3A4
SCHEMBL30464325 0.79 HSD17B10 (0.47) CYP2A6ALDH1A1CYP1A2PRKCZCYP11B2
SCHEMBL10094643 0.77 CYP11B2 (0.54) CYP2A6ALDH1A1CYP1A2PRKCZCYP11B2
SCHEMBL27329360 0.77 HPRT1 (0.54) CYP2A6ALDH1A1CYP1A2TSHRCYP3A4
SCHEMBL10200877 0.76 KDM4E (0.42) ALDH1A1CYP1A2KDM4ECYP3A4CYP2D6
SCHEMBL20873066 0.75 PRKCZ (0.64) CYP1A2PRKCZCYP11B2CYP11B1ADRA2A
SCHEMBL10200876 0.74 KDM4E (0.41) ALDH1A1CYP1A2ADRA2AADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1647 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110818628-B Preparation method of nitrogen-containing aromatic dicarboxylic acid 常熟理工学院 2020-11-06 CN claimed
CN-110818628-A Preparation method of nitrogen-containing aromatic dicarboxylic acid 常熟理工学院 2020-02-21 CN claimed
EP-3542801-A1 PURIN DERIVATIVES FOR USE IN THE TREATMENT OF FAP-RELATED DISEASES Boehringer Ingelheim International GmbH (DE) 2019-09-25 EP claimed
US-20160136180-A1 PURIN DERIVATIVES FOR USE IN THE TREATMENT OF FAB-RELATED DISEASES BOEHRINGER INGELHEIM INT (DE) 2016-05-19 US claimed
US-20110112069-A1 PURIN DERIVATIVES FOR USE IN THE TREATMENT OF FAB-RELATED DISEASES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-05-12 US claimed
CN-101784278-A Purin derivatives for use in the treatment of FAB-related diseases BOEHRINGER INGELHEIM INT 2010-07-21 CN claimed
EP-2190434-A2 PURIN DERIVATIVES FOR USE IN THE TREATMENT OF FAB-RELATED DISEASES Boehringer Ingelheim International GmbH (DE) 2010-06-02 EP claimed
EP-2091929-A1 AGENTS THAT DISRUPT CELLULAR REPLICATION AND THEIR USE IN INHIBITING PATHOLOGICAL CONDITIONS The European Molecular Biology Laboratory (DE) 2009-08-26 EP claimed
WO-2009024542-A2 PURIN DERIVATIVES FOR USE IN THE TREATMENT OF FAB-RELATED DISEASES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-02-26 WO claimed
WO-2007107352-A1 AGENTS THAT DISRUPT CELLULAR REPLICATION AND THEIR USE IN INHIBITING PATHOLOGICAL CONDITIONS THE EUROPEAN MOLECULAR BIOLOGY LABORATORY (DE) 2007-09-27 WO claimed
WO-2024130411-A1 PROTEASE INHIBITORS AND METHODS OF USING SAME VARIATIONAL AI INC. (CA) 2024-06-27 WO disclosed
WO-2024102989-A1 NON-PEPTIDIC SARS-COV-2 MAIN PROTEASE INHIBITORS THE TEXAS A&M UNIVERSITY SYSTEM (US) 2024-05-16 WO disclosed
WO-2024086111-A1 ANTI-VIRAL COMPOUNDS ALIGOS THERAPEUTICS, INC. (US) 2024-04-25 WO disclosed
CN-114907251-B Method for constructing methyl heterocyclic compound by palladium-catalyzed alkyne nucleophilic methylation reaction 大连理工大学 2024-03-08 CN disclosed
CN-114907251-B Method for constructing methyl heterocyclic compound by palladium-catalyzed alkyne nucleophilic methylation reaction 大连理工大学 2024-03-08 CN disclosed
EP-0175263-B1 2-AMINO-3-CHLOROMETHYL-5-(DICHLOROMETHYL)-PYRAZINES AND PROCESS FOR THEIR PREPARATION BASF Aktiengesellschaft (DE) 1991-06-05 EP disclosed
US-4692527-A 2-amino-3,5-di-(halomethyl)-pyrazines and their preparation BASF AKTIENGESELLSCHAFT (DE) 1987-09-08 US disclosed
CN-85102138-A The preparation method of pyrimidoisoquinolinederivatives derivatives 1986-04-10 CN disclosed
EP-0175263-A2 2-Amino-3-chloromethyl-5-(dichloromethyl)-pyrazines and process for their preparation BASF Aktiengesellschaft (DE) 1986-03-26 EP disclosed
US-4053318-A SENSITIZING MEROCYANINE DYE FUJI PHOTO FILM CO., LTD. (JA) 1977-10-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160136180-A1 PURIN DERIVATIVES FOR USE IN THE TREATMENT OF FAB-RELATED DISEASES PNP, ENTPD5, NUDT14 CYP2A6 4497/4885ALDH1A1 3607/4885CYP1A2 4770/4885
US-20110112069-A1 PURIN DERIVATIVES FOR USE IN THE TREATMENT OF FAB-RELATED DISEASES PNP, PURB, NUDT14 CYP2A6 4146/4885ALDH1A1 3774/4885CYP1A2 4692/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.