SCHEMBL4229474

SCHEMBL4229474

OCc1ccc2nc(C(F)(F)F)[nH]c2c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.58
KDM4E B2RXH2 3/20 0.58
HPGD P15428 2/20 0.58
MAPT P10636 2/20 0.58
ALOX15 P16050 2/20 0.58
CYP1A2 P05177 1/20 0.58
CYP2C9 P11712 1/20 0.58
CYP2C19 P33261 1/20 0.58
HSD17B10 Q99714 1/20 0.58
SMN1; SMN2 Q16637 2/20 0.57
NPSR1 Q6W5P4 1/20 0.53
LMNA P02545 2/20 0.52
HTT P42858 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
CBFB Q13951 5/20 0.49
POLB P06746 1/20 0.47
SCN10A Q9Y5Y9 2/20 0.44
KCNH2 Q12809 1/20 0.42
ACP1 P24666 1/20 0.41
NPBWR1 P48145 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9619825 0.87 NPSR1 (0.53) ALDH1A1KDM4EHPGDMAPTALOX15
SCHEMBL26563559 0.84 ALDH1A1 (0.58) ALDH1A1KDM4EHPGDMAPTALOX15
SCHEMBL15110815 0.84 ALDH1A1 (0.58) ALDH1A1KDM4EHPGDMAPTALOX15
SCHEMBL22912817 0.79 KDM4E (0.57) ALDH1A1KDM4EHPGDMAPTALOX15
SCHEMBL6373903 0.79 PKM (0.57) ALDH1A1KDM4EHPGDMAPTALOX15
SCHEMBL29396642 0.79 KDM4E (0.57) ALDH1A1KDM4EHPGDMAPTALOX15
SCHEMBL19970794 0.77 NPBWR1 (0.67) CBFBKCNH2NPBWR1
SCHEMBL10694441 0.76 KDM4E (0.65) ALDH1A1KDM4EHPGDMAPTALOX15
SCHEMBL727388 0.75 PLAU (0.61) ALDH1A1ALOX15CBFBTDP1S1PR1
SCHEMBL6467818 0.75 CBFB (0.52) ALDH1A1ALOX15CYP1A2NPSR1CBFB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2078018-A1 HETEROARYL COMPOUNDS, COMPOSITIONS THEREOF, AND USE THEREOF AS PROTEIN KINASE INHIBITORS Signal Pharmaceuticals LLC (US) 2009-07-15 EP disclosed
WO-2008051494-A1 HETEROARYL COMPOUNDS, COMPOSITIONS THEREOF, AND USE THEREOF AS PROTEIN KINASE INHIBITORS SIGNAL PHARMACEUTICALS, LLC (US) 2008-05-02 WO disclosed