SCHEMBL4229656

SCHEMBL4229656

C[C@@H](N)c1cc(F)cc(C(F)(F)F)c1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 5/20 0.43
PDE2A O00408 1/20 0.40
IDO1 P14902 2/20 0.39
TDO2 P48775 2/20 0.39
CASR P41180 1/20 0.37
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
HTR2B P41595 1/20 0.37
PNMT P11086 1/20 0.36
CACNA1F O60840 1/20 0.35
CACNA1D Q01668 1/20 0.35
CACNA1S Q13698 1/20 0.35
CACNA1C Q13936 1/20 0.35
SOS1 Q07889 2/20 0.33
KRAS P01116 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6819089 1.00 TACR1 (0.43) TACR1PDE2AIDO1TDO2CASR
SCHEMBL336049 0.87 TACR1 (0.51) TACR1PDE2AIDO1TDO2HTR2A
SCHEMBL1728680 0.87 TACR1 (0.51) TACR1PDE2AIDO1TDO2HTR2A
SCHEMBL1492761 0.87 TACR1 (0.51) TACR1PDE2AIDO1TDO2HTR2A
SCHEMBL6917133 0.87 TACR1 (0.51) TACR1PDE2AIDO1TDO2HTR2A
SCHEMBL7939177 0.87 TACR1 (0.51) TACR1PDE2AIDO1TDO2HTR2A
Hydrochloric Acid SCHEMBL7170075 0.85 TACR1 (0.50) TACR1PDE2AIDO1TDO2HTR2A
Hydrochloric Acid SCHEMBL4471353 0.85 TACR1 (0.50) TACR1PDE2AIDO1TDO2HTR2A
Methane SCHEMBL4258949 0.85 TACR1 (0.50) TACR1PDE2AIDO1TDO2HTR2A
Hydrochloric Acid SCHEMBL17439064 0.85 TACR1 (0.50) TACR1PDE2AIDO1TDO2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113727758-A Bicyclic heterocyclic compounds and use thereof 锐新医药公司 2021-11-30 CN disclosed
US-20090099195-A1 Therapeutic Compounds 570 ASTRAZENECA AB (SE) 2009-04-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090099195-A1 Therapeutic Compounds 570 OPRL1, OPRK1, OPRM1 TACR1 16/4885PDE2A 334/4885IDO1 3948/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.