SCHEMBL4230876

SCHEMBL4230876

NC(=O)c1ccc(C(I)c2ccncn2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 1/20 0.39
MKNK1 Q9BUB5 6/20 0.36
MKNK2 Q9HBH9 6/20 0.36
CHEK2 O96017 2/20 0.36
TBXAS1 P24557 1/20 0.35
P2RX7 Q99572 1/20 0.35
TSHR P16473 1/20 0.34
F7 P08709 1/20 0.34
F3 P13726 1/20 0.34
SARM1 Q6SZW1 1/20 0.34
SIRT2 Q8IXJ6 1/20 0.34
SIRT6 Q8N6T7 1/20 0.34
SIRT1 Q96EB6 1/20 0.34
SIRT3 Q9NTG7 1/20 0.34
SIRT5 Q9NXA8 1/20 0.34
SIRT4 Q9Y6E7 1/20 0.34
NNMT P40261 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MAP4K4 O95819 1/20 0.34
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9996419 0.71 NAPRT (0.44) MKNK1MKNK2P2RX7TSHRALDH1A1
SCHEMBL14968784 0.70 P2RX7 (0.43) MKNK1P2RX7TSHRF7F3
SCHEMBL1445286 0.69 MAP4K4 (0.54) CYP17A1MKNK1MKNK2CHEK2MAP4K4
SCHEMBL30251063 0.68 CHEK2 (0.57) CYP17A1MKNK1MKNK2CHEK2TSHR
SCHEMBL2176759 0.68 P2RX7 (0.42) MKNK1P2RX7TSHRSIRT3
SCHEMBL23882643 0.68 CHEK2 (0.57) CYP17A1MKNK1MKNK2CHEK2TSHR
SCHEMBL2176754 0.68 P2RX7 (0.42) MKNK1P2RX7TSHRSIRT3
SCHEMBL23559581 0.67 CYP17A1 (0.49) CYP17A1MKNK1MKNK2CHEK2TSHR
SCHEMBL13434906 0.66 ROCK1 (0.61) MKNK1ROCK1
SCHEMBL4557709 0.66 ALDH1A1 (0.44) P2RX7SMN1; SMN2ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1868611-A4 NOVEL COMPOUNDS GLAXO GROUP LTD (GB) 2009-05-27 EP disclosed
EP-1868611-A2 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2007-12-26 EP disclosed
WO-2006104915-A2 8-PHENYL-7,8-DIHYDROPYRIDO[2,3-d]PYRIMIDIN-7-ONES AND THEIR USE AS PHARMACEUTICALS GLAXO GROUP LIMITED (GB) 2006-10-05 WO disclosed