SCHEMBL4557709

SCHEMBL4557709

NC(=O)C(c1ccccc1)c1ccncn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.44
CYP1A2 P05177 1/20 0.44
HTT P42858 3/20 0.40
GAA P10253 2/20 0.40
CTSD P07339 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
PDGFRA P16234 1/20 0.38
MAPK1 P28482 1/20 0.38
MAPKAPK2 P49137 1/20 0.38
RPS6KA1 Q15418 1/20 0.38
AURKB Q96GD4 1/20 0.38
CSNK1G1 Q9HCP0 1/20 0.38
TDP1 Q9NUW8 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
HDAC4 P56524 2/20 0.37
KDM4E B2RXH2 1/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14968784 0.86 P2RX7 (0.43) CYP1A2CYP3A4TDP1HDAC4KDM4E
SCHEMBL639563 0.81 ALDH1A1 (0.64) ALDH1A1CYP1A2HTTGAACTSD
SCHEMBL7759530 0.81 ALDH1A1 (0.64) ALDH1A1CYP1A2HTTGAACTSD
Hydrochloric Acid SCHEMBL27529639 0.80 ALDH1A1 (0.62) ALDH1A1CYP1A2HTTGAACTSD
Hydrochloric Acid SCHEMBL4200885 0.80 ALDH1A1 (0.62) ALDH1A1CYP1A2HTTGAACTSD
SCHEMBL2205442 0.79 SLC6A2 (0.54) ALDH1A1HTTCTSDMEN1KMT2A
SCHEMBL2492017 0.78 CTSD (0.43) ALDH1A1CYP1A2HTTGAACTSD
SCHEMBL2068072 0.74 HTT (0.43) ALDH1A1CYP1A2HTTGAACTSD
SCHEMBL19664706 0.74 GABBR2 (0.41) ALDH1A1CYP1A2HTTCYP3A4KDM4E
SCHEMBL18426300 0.74 HTT (0.46) ALDH1A1CYP1A2HTTGAACTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009017838-A2 COMBINATIONS OF JAK-2 INHIBITORS AND OTHER AGENTS EXELIXIS, INC. (US) 2009-02-05 WO claimed