SCHEMBL423755

SCHEMBL423755

O=C1CCCN1c1ccc2ncsc2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
L3MBTL1 Q9Y468 3/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
KDM4E B2RXH2 1/20 0.44
HKDC1 Q2TB90 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
HPGD P15428 3/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
CD38 P28907 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
POLB P06746 1/20 0.43
GAA P10253 2/20 0.43
LMNA P02545 1/20 0.43
HTT P42858 1/20 0.43
PIP4K2A P48426 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL413327 0.96 L3MBTL1 (0.43) ALDH1A1L3MBTL1NPC1RAB9AKDM4E
SCHEMBL409024 0.91 LMNA (0.44) ALDH1A1L3MBTL1NPC1RAB9AKDM4E
SCHEMBL410434 0.79 L3MBTL1 (0.45) ALDH1A1L3MBTL1NPC1RAB9AKDM4E
SCHEMBL30688283 0.78 CRBN (0.50) L3MBTL1NPC1RAB9AKDM4EHKDC1
SCHEMBL26683994 0.78 CRBN (0.50) L3MBTL1NPC1RAB9AKDM4EHKDC1
SCHEMBL410875 0.77 CYP3A4 (0.43) L3MBTL1NPC1RAB9AKDM4EHKDC1
SCHEMBL21091414 0.75 GAA (0.57) ALDH1A1L3MBTL1NPC1RAB9AKDM4E
SCHEMBL414419 0.74 DYRK1A (0.42) ALDH1A1L3MBTL1NPC1RAB9AKDM4E
SCHEMBL3785123 0.72 DRD3 (0.44) ALDH1A1L3MBTL1NPC1RAB9AKDM4E
SCHEMBL11142367 0.72 ALDH1A1 (0.74) ALDH1A1L3MBTL1NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2408769-A1 PYRIMIDINE DERIVATIVES USED AS ITK INHIBITORS Glaxo Group Limited (GB) 2012-01-25 EP disclosed
WO-2010106016-A1 PYRIMIDINE DERIVATIVES USED AS ITK INHIBITORS GLAXO GROUP LIMITED (GB) 2010-09-23 WO disclosed