SCHEMBL4239309

SCHEMBL4239309

COC(=O)CCC(C#N)(CCC(=O)OC)c1cccc2c1ccn2C(=O)OCc1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.37
ALDH1A1 P00352 2/20 0.34
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
HTR2C P28335 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
KDM1A O60341 1/20 0.34
MAOA P21397 1/20 0.34
RCOR1 Q9UKL0 1/20 0.34
TACR3 P29371 1/20 0.34
KAT2B Q92831 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
POLB P06746 1/20 0.33
CTSL P07711 2/20 0.32
CTSS P25774 2/20 0.32
CTSB P07858 1/20 0.32
PARP1 P09874 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4239306 0.75 POLB (0.34) ALDH1A1KDM4ELMNASMN1; SMN2POLB
SCHEMBL11821422 0.73 CYP1A2 (0.48) HTTALDH1A1KDM4ETDP1POLB
SCHEMBL29015481 0.73 HTR6 (0.46) ALDH1A1KDM4ELMNAHTR2CKDM1A
SCHEMBL13309267 0.72 NPC1 (0.48) ALDH1A1HTR2CTDP1KDM1AMAOA
SCHEMBL4239275 0.72 TACR3 (0.41) ALDH1A1HTR2CTDP1KDM1AMAOA
SCHEMBL3375069 0.71 TDP1 (0.47) ALDH1A1LMNAHTR2CTDP1KDM1A
SCHEMBL8021561 0.70 ALDH1A1 (0.39) HTTALDH1A1KDM4ELMNARAB9A
SCHEMBL4231904 0.69 TACR3 (0.46) ALDH1A1LMNAHTR2CTDP1KDM1A
SCHEMBL3376524 0.69 KDM1A (0.37) ALDH1A1LMNAHTR2CKDM1AMAOA
SCHEMBL11093234 0.69 ALDH1A1 (0.39) HTTALDH1A1KDM4ELMNATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009115874-A2 NOVEL HETEROCYCLIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESSES FOR THEIR PREPARATION MATRIX LABORATORIES LTD. (IN) 2009-09-24 WO disclosed