SCHEMBL4239559

SCHEMBL4239559

Cc1c(-c2csc(Nc3ccccc3)n2)cnn1-c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLAU P00749 2/20 0.52
RAB9A P51151 7/20 0.50
KMT2A Q03164 5/20 0.50
GAA P10253 4/20 0.50
TRPV4 Q9HBA0 1/20 0.50
MAPT P10636 7/20 0.49
SMN1; SMN2 Q16637 5/20 0.49
NPC1 O15118 5/20 0.49
ALDH1A1 P00352 2/20 0.49
USP2 O75604 1/20 0.49
ALOX15 P16050 1/20 0.49
CLK1 P49759 1/20 0.49
HSD17B10 Q99714 1/20 0.49
MEN1 O00255 4/20 0.48
NFKB1 P19838 3/20 0.48
NFKB2 Q00653 3/20 0.48
RELA Q04206 3/20 0.48
NR1I2 O75469 1/20 0.48
PPP1CA P62136 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4233688 0.94 MEN1 (0.50) PLAURAB9AKMT2AGAATRPV4
SCHEMBL4067193 0.92 VCP (0.57) PLAURAB9AKMT2AGAAMAPT
SCHEMBL12298170 0.92 MAPT (0.54) PLAURAB9AKMT2AGAATRPV4
SCHEMBL4242424 0.92 ALOX5 (0.54) PLAURAB9AKMT2AGAAMAPT
SCHEMBL4065329 0.91 PKM (0.47) PLAURAB9AKMT2AGAATRPV4
SCHEMBL4066150 0.90 PLAU (0.57) PLAURAB9AKMT2AGAATRPV4
SCHEMBL4241367 0.90 AMY1A (0.62) PLAURAB9AKMT2AGAAMAPT
SCHEMBL4057215 0.89 CYP1A2 (0.54) PLAURAB9AKMT2AMAPTSMN1; SMN2
SCHEMBL4243912 0.89 MEN1 (0.52) PLAURAB9AKMT2AGAATRPV4
SCHEMBL4239248 0.87 CFTR (0.56) PLAURAB9AKMT2AMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009010871-A2 PYRAZOLE DERIVATIVES AS ANTAGONISTS OF ADENOSINE A3 RECEPTOR ADDEX PHARMA S.A. (CH) 2009-01-22 WO disclosed