SCHEMBL4241672

SCHEMBL4241672

CN1CCNC(C(=O)c2ccc(-c3ccc(CC4CCN(C5CCCCC5)C4=O)cc3)c(Cl)c2Cl)C1=O

nearest known ligand 0.45

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 2/20 0.45
CES2 O00748 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4241676 0.85 HSD11B1 (0.38) HSD11B1
SCHEMBL4065127 0.82 HSD11B1 (0.58) HSD11B1CES2
SCHEMBL4241674 0.74
SCHEMBL5507886 0.73 HSD11B1 (0.50) HSD11B1CES2
SCHEMBL5511640 0.70 HSD11B1 (0.45) HSD11B1CES2
SCHEMBL3548948 0.69 HSD11B1 (0.74) HSD11B1
SCHEMBL3548392 0.68 HSD11B1 (0.76) HSD11B1CES2
SCHEMBL3542808 0.67 HSD11B1 (0.84) HSD11B1CES2
SCHEMBL4061157 0.67 HSD11B1 (0.47) HSD11B1
SCHEMBL2985349 0.67 HSD11B1 (0.48) HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2016047-A1 BIPHENYL AMIDE LACTAM DERIVATIVES AS INHIBITORS OF 11- BETA-HYDROXYSTEROID DEHYDROGENASE 1 ELI LILLY AND COMPANY (US) 2009-01-21 EP disclosed
WO-2007124337-A1 BIPHENYL AMIDE LACTAM DERIVATIVES AS INHIBITORS OF 11- BETA-HYDROXYSTEROID DEHYDROGENASE 1 ELI LILLY AND COMPANY (US) 2007-11-01 WO disclosed